Abstract
A correlation of in vitro dissolution rate measurements with in vivo pharmacokinetic results in a human study was obtained for a sustained-release formulation of bromocriptine. Different methods were applied to reach this correlation, and the various outcomes were compared.
MeSH terms
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Adult
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Biological Availability
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Blood Pressure / drug effects
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Bromocriptine / administration & dosage
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Bromocriptine / pharmacokinetics*
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Capsules
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Delayed-Action Preparations*
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Half-Life
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Humans
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Male
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Models, Biological
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Pulse / drug effects
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Quality Control
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Solubility
Substances
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Capsules
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Delayed-Action Preparations
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Bromocriptine