Effects of gabaculine, a new potent inhibitor of gamma-amonobutyrate transaminase, on the brain gamma-amonobutyrate content and convulsions in mice

Life Sci. 1977 Apr 1;20(7):1291-5. doi: 10.1016/0024-3205(77)90505-7.
No abstract available

MeSH terms

  • 4-Aminobutyrate Transaminase / antagonists & inhibitors*
  • Aminobutyrates / analysis*
  • Animals
  • Anticonvulsants*
  • Brain Chemistry / drug effects*
  • Cyclohexanecarboxylic Acids / pharmacology*
  • Cyclohexanes / administration & dosage
  • Cyclohexylamines / pharmacology*
  • Dose-Response Relationship, Drug
  • Electroshock
  • Injections, Intraperitoneal
  • Injections, Intraventricular
  • Male
  • Mice
  • Picrotoxin
  • Semicarbazides
  • Time Factors
  • Transaminases / antagonists & inhibitors*
  • gamma-Aminobutyric Acid / analysis*

Substances

  • Aminobutyrates
  • Anticonvulsants
  • Cyclohexanecarboxylic Acids
  • Cyclohexanes
  • Cyclohexylamines
  • Semicarbazides
  • Picrotoxin
  • gabaculine
  • gamma-Aminobutyric Acid
  • Transaminases
  • 4-Aminobutyrate Transaminase