Interaction of SNARE complexes with P/Q-type calcium channels in rat cerebellar synaptosomes

J Biol Chem. 1996 Mar 22;271(12):6567-70. doi: 10.1074/jbc.271.12.6567.

Abstract

P- and Q-type calcium channels, which trigger rapid neurotransmitter release at many mammalian synapses, are blocked by omega-conotoxin MVIIC. 125I-omega-Conotoxin MVIIC binding to rat cerebellar synaptosomes was not displaced by omega-conotoxins GVIA or MVIIA (Ki > 1 microM), which are selective for N-type calcium channels. Solubilized 125I-omega-conotoxin MVIIC receptors were specifically recognized by antibodies directed against alpha1A calcium channel subunits, proteins known to constitute a pore with P/Q-like channel properties. Antibodies against syntaxin 1, SNAP 25, and VAMP 2 (synaptobrevin) each immunoprecipitated a similar fraction (20-40%) of omega-conotoxin MVIIC receptors. Immunoprecipitation was not additive, suggesting that heterotrimeric (SNARE) complexes containing these three proteins interact with P/Q-type calcium channels. Immobilized monoclonal anti-syntaxin antibodies retained alpha1A calcium channel subunits of 220, 180 and 160 kDa monitored by immunoblotting with site directed antibodies. Synaptotagmin was detected in channel-associated complexes, but not synaptophysin, Rab 3A nor rat cysteine string protein. Trimeric SNARE complexes are implicated in calcium-dependent exocytosis, a process thought to be regulated by synaptotagmin. Our results indicate that these proteins interact with P/Q-type calcium channels, which may optimize their location within domains of calcium influx.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium Channel Blockers / chemistry
  • Calcium Channel Blockers / metabolism
  • Calcium Channels / chemistry
  • Calcium Channels / metabolism*
  • Cerebellum / metabolism*
  • Membrane Proteins / metabolism*
  • Molecular Probes
  • Mollusk Venoms / chemistry
  • Mollusk Venoms / metabolism
  • Protein Binding
  • Rats
  • SNARE Proteins
  • Synaptosomes / metabolism*
  • Syntaxin 1
  • Vesicular Transport Proteins*

Substances

  • Calcium Channel Blockers
  • Calcium Channels
  • Membrane Proteins
  • Molecular Probes
  • Mollusk Venoms
  • SNARE Proteins
  • Stx1a protein, rat
  • Syntaxin 1
  • Vesicular Transport Proteins