[Synthesis and pharmacological study of various 2-(alkylaminoalkyl)mercapto-5-aryl-1,3,4-oxadiazoles]

Farmaco Sci. 1977 Jun;32(6):414-29.
[Article in Italian]

Abstract

Work was continued on the pharmacological study of the 1,3,4-oxadiazole nucleus using aroylhydrazines already used for the synthesis of anti-MAO compounds. S-alkylaminoalkyl derivatives of some 2-mercapto-5-aryl-1,3,4-oxadiazoles were prepared bearing in the 5-position a 3,4,5-trimethoxyphenyl, a 3,5-dimethoxy-4-ethoxyphenyl or a 3,4-dihydroxymethylenephenyl radical. When subjected to pharmacological investigation the compounds showed clear hypotensive activity partially antagonized by atropine and antispastic activity on smooth muscle.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Antihypertensive Agents / chemical synthesis*
  • Blood Pressure / drug effects
  • Chemical Phenomena
  • Chemistry
  • Guinea Pigs
  • Ileum / drug effects
  • Male
  • Mice
  • Muscle, Smooth / drug effects
  • Oxadiazoles / chemical synthesis*
  • Oxadiazoles / pharmacology
  • Rabbits
  • Rats

Substances

  • Antihypertensive Agents
  • Oxadiazoles