Maintenance of growth factor signaling through Ras in human colon carcinoma cells containing K-ras mutations

Int J Cancer. 1996 Aug 7;67(4):539-46. doi: 10.1002/(SICI)1097-0215(19960807)67:4<539::AID-IJC13>3.0.CO;2-2.

Abstract

Fifty percent of human colon carcinomas contain activating mutations in the K-ras gene. However, whether these alterations in K-ras affect the function of Ras proteins in growth factor (GF) signal transduction is now known. Here we have characterized a previously defined human colon carcinoma cell model system for K-ras gene mutations and for altered levels of Ras protein expression and have examined whether these alterations affect Ras function in GF signal transduction. Sequence analysis of PCR-amplified K-ras gene fragments indicated that among the more aggressive cell lines, four had a normal K-ras sequence, whereas 3 others (isolated from the same human tumor) contained a mutation at codon 13. In contrast, all 7 of the less aggressive cell lines contained a mutation at either codon 12 or 13. In addition to the presence of a K-ras mutation, one cell line expressed higher levels of the K-Ras protein and displayed elevated Ras-GTP loading (in the absence of GF addition) compared with the other cell lines examined. Despite these alterations, the mitogenic GF combination epidermal growth factor + insulin + transferrin resulted in an activation of Ras and extracellular signal-regulated kinase 2. Collectively, our results indicate that the malignant phenotype of the cell lines was not correlated with the presence of K-ras mutations or with higher levels of Ras protein expression. Furthermore, K-ras mutations, high levels of K-Ras protein expression, and elevated Ras-GTP loading, as they occur naturally in human colon carcinomas, do not abolish the function of Ras in GF signaling.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Base Sequence
  • Blotting, Western
  • Cell Line
  • Codon
  • Colonic Neoplasms
  • DNA Primers
  • Epidermal Growth Factor / pharmacology
  • Exons
  • Genes, ras*
  • Growth Substances / pharmacology*
  • Guanosine Triphosphate / metabolism
  • Humans
  • Insulin / pharmacology
  • Kinetics
  • Molecular Sequence Data
  • Point Mutation*
  • Polymerase Chain Reaction
  • Signal Transduction*
  • Transferrin / pharmacology
  • Tumor Cells, Cultured
  • ras Proteins / biosynthesis
  • ras Proteins / physiology*

Substances

  • Codon
  • DNA Primers
  • Growth Substances
  • Insulin
  • Transferrin
  • Epidermal Growth Factor
  • Guanosine Triphosphate
  • ras Proteins