Genetic evidence for involvement of type 1, type 2 and type 3 inositol 1,4,5-trisphosphate receptors in signal transduction through the B-cell antigen receptor

EMBO J. 1997 Jun 2;16(11):3078-88. doi: 10.1093/emboj/16.11.3078.

Abstract

Stimulation of B-cell antigen receptor (BCR) induces a rapid increase in cytoplasmic free calcium due to its release from intracellular stores and influx from the extracellular environment. Inositol 1,4,5-trisphosphate receptors (IP3Rs) are ligand-gated channels that release intracellular calcium stores in response to the second messenger, inositol 1,4,5-trisphosphate. Most hematopoietic cells, including B cells, express at least two of the three different types of IP3R. We demonstrate here that B cells in which a single type of IP3R has been deleted still mobilize calcium in response to BCR stimulation, whereas this calcium mobilization is abrogated in B cells lacking all three types of IP3R. Calcium mobilization by a transfected G protein-coupled receptor (muscarinic M1 receptor) was also abolished in only triple-deficient cells. Capacitative Ca2+ entry, stimulated by thapsigargin, remains unaffected by loss of all three types of IP3R. These data establish that IP3Rs are essential and functionally redundant mediators for both BCR- and muscarinic receptor-induced calcium mobilization, but not for thapsigargin-induced Ca2+ influx. We further show that the BCR-induced apoptosis is significantly inhibited by loss of all three types of IP3R, suggesting an important role for Ca2+ in the process of apoptosis.

MeSH terms

  • Biological Transport
  • Calcium / metabolism
  • Calcium Channels / classification
  • Calcium Channels / genetics
  • Calcium Channels / metabolism*
  • Cell Line
  • Enzyme Activation
  • Inositol 1,4,5-Trisphosphate / metabolism*
  • Inositol 1,4,5-Trisphosphate Receptors
  • Intracellular Signaling Peptides and Proteins*
  • Isoenzymes / metabolism
  • Membrane Proteins*
  • Mutation
  • Myristoylated Alanine-Rich C Kinase Substrate
  • Phospholipase C gamma
  • Proteins / metabolism
  • Receptor, Muscarinic M1
  • Receptors, Antigen, B-Cell / metabolism*
  • Receptors, Cytoplasmic and Nuclear / classification
  • Receptors, Cytoplasmic and Nuclear / genetics
  • Receptors, Cytoplasmic and Nuclear / metabolism*
  • Receptors, Muscarinic / metabolism
  • Signal Transduction*
  • Thapsigargin / pharmacology
  • Type C Phospholipases / metabolism

Substances

  • Calcium Channels
  • Inositol 1,4,5-Trisphosphate Receptors
  • Intracellular Signaling Peptides and Proteins
  • Isoenzymes
  • Membrane Proteins
  • Proteins
  • Receptor, Muscarinic M1
  • Receptors, Antigen, B-Cell
  • Receptors, Cytoplasmic and Nuclear
  • Receptors, Muscarinic
  • Myristoylated Alanine-Rich C Kinase Substrate
  • Thapsigargin
  • Inositol 1,4,5-Trisphosphate
  • Type C Phospholipases
  • Phospholipase C gamma
  • Calcium