Inhibition of acetylcholine esterase and choline esterase by benzethonium chloride and avoidance of the benzethonium chloride carry-over inhibitory effect

Eur J Clin Chem Clin Biochem. 1997 Aug;35(8):603-7. doi: 10.1515/cclm.1997.35.8.603.

Abstract

It has been shown that benzethonium chloride produces linear mixed-type inhibition of choline esterase and acetylcholine esterase. These enzymes also show-reagent-carry-over inhibition if the enzyme activities are measured in plastic cuvettes in which previously protein has been determined by the alkaline benzethonium chloride method. Choline esterase is about 10-fold more sensitive to benzethonium chloride than acetylcholine esterase. With acetylthiocholine as substrate Michaelis-Menten constants for choline esterase and acetylcholine esterase are 85 mumol/l and 102 mumol/l, respectively. Carry-over inhibitory effect of benzethonium chloride can be avoided by washing the cuvettes, after protein determination by the benzethonium chloride method, with 5 ml/l Triton X-100, 5 ml/l Tween 20 or 10 g/l sodium dodecyl sulphate. The latter has a disadvantage in that it precipitates out at low temperatures. The dry slide method (Johnson & Johnson) for serum choline esterase is free of the inhibitory effect until the concentration of benzethonium chloride in the sample reaches about 200 mumol/l.

MeSH terms

  • Acetylcholinesterase / drug effects*
  • Acetylcholinesterase / metabolism
  • Benzethonium / adverse effects
  • Benzethonium / pharmacology*
  • Butyrylthiocholine / metabolism
  • Cholinesterase Inhibitors / adverse effects
  • Cholinesterase Inhibitors / pharmacology*
  • Cholinesterases / drug effects*
  • Cholinesterases / metabolism
  • Humans
  • Indicators and Reagents / adverse effects
  • Kinetics
  • Substrate Specificity

Substances

  • Cholinesterase Inhibitors
  • Indicators and Reagents
  • Benzethonium
  • Butyrylthiocholine
  • Acetylcholinesterase
  • Cholinesterases