Characterization of two polyubiquitin binding sites in the 26 S protease subunit 5a

J Biol Chem. 1998 Mar 6;273(10):5461-7. doi: 10.1074/jbc.273.10.5461.

Abstract

Ubiquitylated proteins are degraded by the 26 S protease, an enzyme complex that contains 30 or more unique subunits. One of these proteins, subunit 5a (S5a), has been shown to bind ubiquitin-lysozyme conjugates and free polyubiquitin chains. Using deletional analysis, we have identified in the carboxyl-terminal half of human S5a, two independent polyubiquitin binding sites whose sequences are highly conserved among higher eukaryotic S5a homologs. The sites are approximately 30-amino acids long and are separated by 50 intervening residues. When expressed as small fragments or when present in full-length S5a molecules, the sites differ at least 10-fold in their apparent affinity for polyubiquitin chains. Each binding site contains 5 hydrophobic residues that form an alternating pattern of large and small side chains, e.g. Leu-Ala-Leu-Ala-Leu, and this pattern is essential for binding ubiquitin chains. Based on the importance of the alternating hydrophobic residues in the binding sites and previous studies showing that a hydrophobic patch on the surface of ubiquitin is essential for proteolytic targeting, we propose a model for molecular recognition of polyubiquitin chains by S5a.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Binding Sites / physiology
  • Biopolymers / metabolism*
  • Conserved Sequence / genetics
  • Humans
  • Molecular Sequence Data
  • Muramidase / metabolism
  • Mutagenesis, Site-Directed / genetics
  • Peptide Fragments / chemistry
  • Peptide Fragments / pharmacology
  • Peptide Hydrolases / chemistry*
  • Peptide Hydrolases / physiology
  • Polyubiquitin
  • Proteasome Endopeptidase Complex*
  • Protein Binding / physiology
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / pharmacology
  • Sequence Deletion / genetics
  • Sequence Homology, Amino Acid
  • Ubiquitins / metabolism*

Substances

  • Biopolymers
  • Peptide Fragments
  • Recombinant Proteins
  • Ubiquitins
  • Polyubiquitin
  • Muramidase
  • Peptide Hydrolases
  • Proteasome Endopeptidase Complex
  • ATP dependent 26S protease