Regulation of levels of 5-HT2A receptor mRNA

Ann N Y Acad Sci. 1998 Dec 15:861:128-35. doi: 10.1111/j.1749-6632.1998.tb10183.x.

Abstract

We have been able to identify two separate pathways present in P11 cells that can increase the levels and stability of 5-HT2A receptor mRNA. One pathway is activated following exposure of cells to serotonin and is dependent upon activation of a PKC isoform that is susceptible to downregulation by a 24-h pretreatment with PMA; another pathway is activated following treatment of cells with a calcium ionophore. This pathway is not dependent on activation of PKC isoforms that can be downregulated by a 24-h treatment with phorbol ester. Such heterologous regulation of levels of 5-HT2A receptor mRNA may be important in understanding in vivo events where multiple factors contribute to the modulation of levels of cell surface receptors.

Publication types

  • Review

MeSH terms

  • Animals
  • Brain / metabolism*
  • Female
  • Gene Expression Regulation* / drug effects
  • Models, Biological
  • Myometrium / metabolism
  • RNA, Messenger / genetics
  • Receptor, Serotonin, 5-HT2A
  • Receptors, Serotonin / genetics*
  • Serotonin Antagonists / pharmacology
  • Serotonin Receptor Agonists / pharmacology
  • Signal Transduction
  • Transcription, Genetic* / drug effects

Substances

  • RNA, Messenger
  • Receptor, Serotonin, 5-HT2A
  • Receptors, Serotonin
  • Serotonin Antagonists
  • Serotonin Receptor Agonists