Discovery of a Potent SARM1 Base-Exchange Inhibitor with In Vivo Efficacy.
Giroud M, Kuhn B, Steiner S, Westwood P, Mendel M, Mani A, Pinard E, Haap W, Grether U, Caramenti P, Rombach D, Zambaldo C, Ritter M, Schmid P, Gasser C, Aregger N, Séchet N, Topp A, Bilyard M, Malnight-Alvarez A, Plitzko I, Hilbert M, Kalayil S, Burger D, Bonardi C, Saal W, Haider A, Wittwer MB, Brigo A, Benz J, Keaney J.
Giroud M, et al. Among authors: haider a.
J Med Chem. 2025 Mar 27;68(6):6558-6575. doi: 10.1021/acs.jmedchem.4c03127. Epub 2025 Mar 18.
J Med Chem. 2025.
PMID: 40100796