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Year Number of Results
2004 1
2006 1
2007 1
2011 1
2012 1
2013 1
2014 1
2015 1
2017 2
2018 1
2019 5
2020 4
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Page 1
Contribution of Pretomanid to Novel Regimens Containing Bedaquiline with either Linezolid or Moxifloxacin and Pyrazinamide in Murine Models of Tuberculosis.
Xu J, Li SY, Almeida DV, Tasneen R, Barnes-Boyle K, Converse PJ, Upton AM, Mdluli K, Fotouhi N, Nuermberger EL. Xu J, et al. Among authors: upton am. Antimicrob Agents Chemother. 2019 Apr 25;63(5):e00021-19. doi: 10.1128/AAC.00021-19. Print 2019 May. Antimicrob Agents Chemother. 2019. PMID: 30833432 Free PMC article.
Structure-activity relationships for analogs of the tuberculosis drug bedaquiline with the naphthalene unit replaced by bicyclic heterocycles.
Sutherland HS, Tong AST, Choi PJ, Conole D, Blaser A, Franzblau SG, Cooper CB, Upton AM, Lotlikar MU, Denny WA, Palmer BD. Sutherland HS, et al. Among authors: upton am. Bioorg Med Chem. 2018 May 1;26(8):1797-1809. doi: 10.1016/j.bmc.2018.02.026. Epub 2018 Feb 20. Bioorg Med Chem. 2018. PMID: 29482950 Free PMC article.
3,5-Dialkoxypyridine analogues of bedaquiline are potent antituberculosis agents with minimal inhibition of the hERG channel.
Sutherland HS, Tong AST, Choi PJ, Blaser A, Conole D, Franzblau SG, Lotlikar MU, Cooper CB, Upton AM, Denny WA, Palmer BD. Sutherland HS, et al. Among authors: upton am. Bioorg Med Chem. 2019 Apr 1;27(7):1292-1307. doi: 10.1016/j.bmc.2019.02.026. Epub 2019 Feb 15. Bioorg Med Chem. 2019. PMID: 30803745 Free PMC article.
Variations in the C-unit of bedaquiline provides analogues with improved biology and pharmacology.
Sutherland HS, Tong AST, Choi PJ, Blaser A, Franzblau SG, Cooper CB, Upton AM, Lotlikar M, Denny WA, Palmer BD. Sutherland HS, et al. Among authors: upton am. Bioorg Med Chem. 2020 Jan 1;28(1):115213. doi: 10.1016/j.bmc.2019.115213. Epub 2019 Nov 26. Bioorg Med Chem. 2020. PMID: 31810890
Structure-activity relationships for unit C pyridyl analogues of the tuberculosis drug bedaquiline.
Blaser A, Sutherland HS, Tong AST, Choi PJ, Conole D, Franzblau SG, Cooper CB, Upton AM, Lotlikar M, Denny WA, Palmer BD. Blaser A, et al. Among authors: upton am. Bioorg Med Chem. 2019 Apr 1;27(7):1283-1291. doi: 10.1016/j.bmc.2019.02.025. Epub 2019 Feb 15. Bioorg Med Chem. 2019. PMID: 30792104 Free PMC article.
6-Cyano Analogues of Bedaquiline as Less Lipophilic and Potentially Safer Diarylquinolines for Tuberculosis.
Tong AST, Choi PJ, Blaser A, Sutherland HS, Tsang SKY, Guillemont J, Motte M, Cooper CB, Andries K, Van den Broeck W, Franzblau SG, Upton AM, Denny WA, Palmer BD, Conole D. Tong AST, et al. Among authors: upton am. ACS Med Chem Lett. 2017 Sep 22;8(10):1019-1024. doi: 10.1021/acsmedchemlett.7b00196. eCollection 2017 Oct 12. ACS Med Chem Lett. 2017. PMID: 29057044 Free PMC article.
Synthesis and evaluation of analogues of the tuberculosis drug bedaquiline containing heterocyclic B-ring units.
Choi PJ, Sutherland HS, Tong AST, Blaser A, Franzblau SG, Cooper CB, Lotlikar MU, Upton AM, Guillemont J, Motte M, Queguiner L, Andries K, Van den Broeck W, Denny WA, Palmer BD. Choi PJ, et al. Among authors: upton am. Bioorg Med Chem Lett. 2017 Dec 1;27(23):5190-5196. doi: 10.1016/j.bmcl.2017.10.042. Epub 2017 Oct 20. Bioorg Med Chem Lett. 2017. PMID: 29107541 Free PMC article.
TBAJ-876 Retains Bedaquiline's Activity against Subunits c and ε of Mycobacterium tuberculosis F-ATP Synthase.
Sarathy JP, Ragunathan P, Shin J, Cooper CB, Upton AM, Grüber G, Dick T. Sarathy JP, et al. Among authors: upton am. Antimicrob Agents Chemother. 2019 Sep 23;63(10):e01191-19. doi: 10.1128/AAC.01191-19. Print 2019 Oct. Antimicrob Agents Chemother. 2019. PMID: 31358589 Free PMC article.
Synergistic Activity of Nitroimidazole-Oxazolidinone Conjugates against Anaerobic Bacteria.
Zhuang Z, Wan D, Ding J, He S, Zhang Q, Wang X, Yuan Y, Lu Y, Ding CZ, Lynch AS, Upton AM, Cooper CB, Denny WA, Ma Z. Zhuang Z, et al. Among authors: upton am. Molecules. 2020 May 22;25(10):2431. doi: 10.3390/molecules25102431. Molecules. 2020. PMID: 32456032 Free PMC article.
TBAJ-876 Displays Bedaquiline-Like Mycobactericidal Potency without Retaining the Parental Drug's Uncoupler Activity.
Sarathy JP, Ragunathan P, Cooper CB, Upton AM, Grüber G, Dick T. Sarathy JP, et al. Among authors: upton am. Antimicrob Agents Chemother. 2020 Jan 27;64(2):e01540-19. doi: 10.1128/AAC.01540-19. Print 2020 Jan 27. Antimicrob Agents Chemother. 2020. PMID: 31712198 Free PMC article.
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