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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
2003 1
2006 2
2007 1
2008 2
2009 2
2010 1
2014 1
2015 2
2016 4
2017 1
2018 1
2019 1
2020 0
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18 results
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Page 1
Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4-f]quinazolin-9(8H)-one, a Promising Inhibitor of DYRK1A.
Fruit C, Couly F, Bhansali R, Rammohan M, Lindberg MF, Crispino JD, Meijer L, Besson T. Fruit C, et al. Pharmaceuticals (Basel). 2019 Dec 17;12(4):185. doi: 10.3390/ph12040185. Pharmaceuticals (Basel). 2019. PMID: 31861110 Free PMC article.
Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors: a survey of recent patent literature.
Nguyen TL, Fruit C, Hérault Y, Meijer L, Besson T. Nguyen TL, et al. Among authors: fruit c. Expert Opin Ther Pat. 2017 Nov;27(11):1183-1199. doi: 10.1080/13543776.2017.1360285. Epub 2017 Aug 2. Expert Opin Ther Pat. 2017. PMID: 28766366 Review.
Development of Kinase Inhibitors via Metal-Catalyzed C⁻H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies.
Couly F, Harari M, Dubouilh-Benard C, Bailly L, Petit E, Diharce J, Bonnet P, Meijer L, Fruit C, Besson T. Couly F, et al. Among authors: fruit c. Molecules. 2018 Aug 29;23(9):2181. doi: 10.3390/molecules23092181. Molecules. 2018. PMID: 30158487 Free PMC article.
Aminoacid-derived mercaptoimidazoles.
Crépin A, Wattier N, Petit S, Bischoff L, Fruit C, Marsais F. Crépin A, et al. Among authors: fruit c. Org Biomol Chem. 2009 Jan 7;7(1):128-34. doi: 10.1039/b810678a. Epub 2008 Oct 31. Org Biomol Chem. 2009. PMID: 19081955
Synthesis of Bioactive 2-(Arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff Reaction or Cu- Catalyzed Intramolecular C-S Bond Formation.
Hédou D, Dubouilh-Benard C, Loaëc N, Meijer L, Fruit C, Besson T. Hédou D, et al. Among authors: fruit c. Molecules. 2016 Jun 18;21(6):794. doi: 10.3390/molecules21060794. Molecules. 2016. PMID: 27322235 Free PMC article.
ORGANIC CHEMISTRY. Three catalysts for activating carbon-hydrogen bonds.
Fruit C. Fruit C. Science. 2016 Jun 10;352(6291):1277-8. doi: 10.1126/science.aaf8923. Science. 2016. PMID: 27284182 No abstract available.
Ligand-free Pd-catalyzed and copper-assisted C-H arylation of quinazolin-4-ones with aryl iodides under microwave heating.
Laclef S, Harari M, Godeau J, Schmitz-Afonso I, Bischoff L, Hoarau C, Levacher V, Fruit C, Besson T. Laclef S, et al. Among authors: fruit c. Org Lett. 2015 Apr 3;17(7):1700-3. doi: 10.1021/acs.orglett.5b00467. Epub 2015 Mar 17. Org Lett. 2015. PMID: 25781369
Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides.
Harari M, Couly F, Fruit C, Besson T. Harari M, et al. Among authors: fruit c. Org Lett. 2016 Jul 1;18(13):3282-5. doi: 10.1021/acs.orglett.6b01552. Epub 2016 Jun 17. Org Lett. 2016. PMID: 27314437
Regioselective decarboxylative cross-coupling of carboxy isoquinoline N-oxides.
Rouchet JB, Schneider C, Fruit C, Hoarau C. Rouchet JB, et al. Among authors: fruit c. J Org Chem. 2015 Jun 5;80(11):5919-27. doi: 10.1021/acs.joc.5b00475. Epub 2015 May 14. J Org Chem. 2015. PMID: 25938169
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