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Year Number of Results
2011 1
2012 1
2013 3
2014 5
2015 3
2016 2
2017 3
2018 3
2019 1
2020 2
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22 results
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Page 1
Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants.
Marek M, Shaik TB, Heimburg T, Chakrabarti A, Lancelot J, Ramos-Morales E, Da Veiga C, Kalinin D, Melesina J, Robaa D, Schmidtkunz K, Suzuki T, Holl R, Ennifar E, Pierce RJ, Jung M, Sippl W, Romier C. Marek M, et al. Among authors: lancelot j. J Med Chem. 2018 Nov 21;61(22):10000-10016. doi: 10.1021/acs.jmedchem.8b01087. Epub 2018 Nov 8. J Med Chem. 2018. PMID: 30347148
Structure-Reactivity Relationships on Substrates and Inhibitors of the Lysine Deacylase Sirtuin 2 from Schistosoma mansoni (SmSirt2).
Monaldi D, Rotili D, Lancelot J, Marek M, Wössner N, Lucidi A, Tomaselli D, Ramos-Morales E, Romier C, Pierce RJ, Mai A, Jung M. Monaldi D, et al. Among authors: lancelot j. J Med Chem. 2019 Oct 10;62(19):8733-8759. doi: 10.1021/acs.jmedchem.9b00638. Epub 2019 Sep 20. J Med Chem. 2019. PMID: 31496251
Schistosome sirtuins as drug targets.
Lancelot J, Cabezas-Cruz A, Caby S, Marek M, Schultz J, Romier C, Sippl W, Jung M, Pierce RJ. Lancelot J, et al. Future Med Chem. 2015;7(6):765-82. doi: 10.4155/fmc.15.24. Future Med Chem. 2015. PMID: 25996069 Free article. Review.
Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as SmHDAC8 Inhibitors for the Treatment of Schistosomiasis.
Bayer T, Chakrabarti A, Lancelot J, Shaik TB, Hausmann K, Melesina J, Schmidtkunz K, Marek M, Erdmann F, Schmidt M, Robaa D, Romier C, Pierce RJ, Jung M, Sippl W. Bayer T, et al. Among authors: lancelot j. ChemMedChem. 2018 Aug 10;13(15):1517-1529. doi: 10.1002/cmdc.201800238. Epub 2018 Jul 4. ChemMedChem. 2018. PMID: 29806110
Epigenetic control of gene function in schistosomes: a source of therapeutic targets?
Cabezas-Cruz A, Lancelot J, Caby S, Oliveira G, Pierce RJ. Cabezas-Cruz A, et al. Among authors: lancelot j. Front Genet. 2014 Sep 10;5:317. doi: 10.3389/fgene.2014.00317. eCollection 2014. Front Genet. 2014. PMID: 25309576 Free PMC article. Review.
A Novel Class of Schistosoma mansoni Histone Deacetylase 8 (HDAC8) Inhibitors Identified by Structure-Based Virtual Screening and In Vitro Testing.
Simoben CV, Robaa D, Chakrabarti A, Schmidtkunz K, Marek M, Lancelot J, Kannan S, Melesina J, Shaik TB, Pierce RJ, Romier C, Jung M, Sippl W. Simoben CV, et al. Among authors: lancelot j. Molecules. 2018 Mar 2;23(3):566. doi: 10.3390/molecules23030566. Molecules. 2018. PMID: 29498707 Free PMC article.
Targeting schistosome histone modifying enzymes for drug development.
Pierce RJ, Dubois-Abdesselem F, Lancelot J, Andrade L, Oliveira G. Pierce RJ, et al. Among authors: lancelot j. Curr Pharm Des. 2012;18(24):3567-78. Curr Pharm Des. 2012. PMID: 22607147 Review.
Isophthalic Acid-Based HDAC Inhibitors as Potent Inhibitors of HDAC8 from Schistosoma mansoni.
Stenzel K, Chakrabarti A, Melesina J, Hansen FK, Lancelot J, Herkenhöhner S, Lungerich B, Marek M, Romier C, Pierce RJ, Sippl W, Jung M, Kurz T. Stenzel K, et al. Among authors: lancelot j. Arch Pharm (Weinheim). 2017 Aug;350(8). doi: 10.1002/ardp.201700096. Epub 2017 Jun 22. Arch Pharm (Weinheim). 2017. PMID: 28639720
Analysis of the interactome of Schistosoma mansoni histone deacetylase 8.
Caby S, Pagliazzo L, Lancelot J, Saliou JM, Bertheaume N, Pierce RJ, Roger E. Caby S, et al. Among authors: lancelot j. PLoS Negl Trop Dis. 2017 Nov 20;11(11):e0006089. doi: 10.1371/journal.pntd.0006089. eCollection 2017 Nov. PLoS Negl Trop Dis. 2017. PMID: 29155817 Free PMC article.
Effect of clinically approved HDAC inhibitors on Plasmodium, Leishmania and Schistosoma parasite growth.
Chua MJ, Arnold MS, Xu W, Lancelot J, Lamotte S, Späth GF, Prina E, Pierce RJ, Fairlie DP, Skinner-Adams TS, Andrews KT. Chua MJ, et al. Among authors: lancelot j. Int J Parasitol Drugs Drug Resist. 2017 Apr;7(1):42-50. doi: 10.1016/j.ijpddr.2016.12.005. Epub 2016 Dec 23. Int J Parasitol Drugs Drug Resist. 2017. PMID: 28107750 Free PMC article.
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