Malken Bayrakdarian - Search Results

Year	Number of Results
2002	2
2005	3
2006	1
2008	1
2009	1
2011	1
2012	1
2014	1
2018	1
2025	1
2026	0

1

Radiolabeling and Preliminary In Vivo Evaluation of the Candidate CCR2 Targeting PET Radioligand [¹¹C]AZD2423.

Dahl K, Johnström P, Tóth M, Bolin M, Varnäs K, Nakao R, Takano A, Khani Meynaq Y, Bayrakdarian M, Cselényi Z, Halldin C, Farde L, Schou M. Dahl K, et al. Among authors: bayrakdarian m. Pharmaceuticals (Basel). 2025 Jan 21;18(2):135. doi: 10.3390/ph18020135. Pharmaceuticals (Basel). 2025. PMID: 40005950 Free PMC article.

2

Discovery of P2X3 selective antagonists for the treatment of chronic pain.

Cantin LD, Bayrakdarian M, Buon C, Grazzini E, Hu YJ, Labrecque J, Leung C, Luo X, Martino G, Paré M, Payza K, Popovic N, Projean D, Santhakumar V, Walpole C, Yu XH, Tomaszewski MJ. Cantin LD, et al. Among authors: bayrakdarian m. Bioorg Med Chem Lett. 2012 Apr 1;22(7):2565-71. doi: 10.1016/j.bmcl.2012.01.124. Epub 2012 Feb 9. Bioorg Med Chem Lett. 2012. PMID: 22370269

3

Discovery and pharmacological characterization of a small-molecule antagonist at neuromedin U receptor NMUR2.

Liu JJ, Payza K, Huang J, Liu R, Chen T, Coupal M, Laird JM, Cao CQ, Butterworth J, Lapointe S, Bayrakdarian M, Trivedi S, Bostwick JR. Liu JJ, et al. Among authors: bayrakdarian m. J Pharmacol Exp Ther. 2009 Jul;330(1):268-75. doi: 10.1124/jpet.109.152967. Epub 2009 Apr 15. J Pharmacol Exp Ther. 2009. PMID: 19369576

4

Asymmetric Synthesis of a Potent CXCR7 Modulator Featuring a Hindered Tertiary β-Amino Amide Stereocenter.

Canterbury DP, Godin F, Desjardins S, Bayrakdarian M, Albert JS, Perry DA, Hesp KD. Canterbury DP, et al. Among authors: bayrakdarian m. Org Lett. 2018 Sep 7;20(17):5336-5339. doi: 10.1021/acs.orglett.8b02261. Epub 2018 Aug 17. Org Lett. 2018. PMID: 30118238

5

Total synthesis of A-315675: a potent inhibitor of influenza neuraminidase.

Hanessian S, Bayrakdarian M, Luo X. Hanessian S, et al. Among authors: bayrakdarian m. J Am Chem Soc. 2002 May 1;124(17):4716-21. doi: 10.1021/ja0126226. J Am Chem Soc. 2002. PMID: 11971721

6

Development of 2,4-diaminopyrimidine derivatives as novel SNSR4 antagonists.

Bayrakdarian M, Butterworth J, Hu YJ, Santhakumar V, Tomaszewski MJ. Bayrakdarian M, et al. Bioorg Med Chem Lett. 2011 Apr 1;21(7):2102-5. doi: 10.1016/j.bmcl.2011.01.138. Epub 2011 Feb 3. Bioorg Med Chem Lett. 2011. PMID: 21333534

7

Phenolic P2/P3 core motif as thrombin inhibitors--design, synthesis, and X-ray co-crystal structure.

Hanessian S, Therrien E, van Otterlo WA, Bayrakdarian M, Nilsson I, Fjellström O, Xue Y. Hanessian S, et al. Among authors: bayrakdarian m. Bioorg Med Chem Lett. 2006 Feb 15;16(4):1032-6. doi: 10.1016/j.bmcl.2005.10.082. Epub 2005 Nov 15. Bioorg Med Chem Lett. 2006. PMID: 16290930

8

Structure-based design, synthesis, and memapsin 2 (BACE) inhibitory activity of carbocyclic and heterocyclic peptidomimetics.

Hanessian S, Yun H, Hou Y, Yang G, Bayrakdarian M, Therrien E, Moitessier N, Roggo S, Veenstra S, Tintelnot-Blomley M, Rondeau JM, Ostermeier C, Strauss A, Ramage P, Paganetti P, Neumann U, Betschart C. Hanessian S, et al. Among authors: bayrakdarian m. J Med Chem. 2005 Aug 11;48(16):5175-90. doi: 10.1021/jm050142+. J Med Chem. 2005. PMID: 16078837

9

Design and synthesis of a novel class of constrained tricyclic pyrrolizidinone carboxylic acids as carbapenem mimics.

Hanessian S, Buckle R, Bayrakdarian M. Hanessian S, et al. Among authors: bayrakdarian m. J Org Chem. 2002 May 17;67(10):3387-97. doi: 10.1021/jo0111715. J Org Chem. 2002. PMID: 12003550

10

Reactive metabolite trapping screens and potential pitfalls: bioactivation of a homomorpholine and formation of an unstable thiazolidine adduct.

Lenz EM, Martin S, Schmidt R, Morin PE, Smith R, Weston DJ, Bayrakdarian M. Lenz EM, et al. Among authors: bayrakdarian m. Chem Res Toxicol. 2014 Jun 16;27(6):968-80. doi: 10.1021/tx5000409. Epub 2014 Jun 5. Chem Res Toxicol. 2014. PMID: 24855970

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Results by year

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

12 results

Results by year

Search Page

Filters

My Custom Filters

Results by year

Publication date

Text availability

Article attribute

Article type

Additional filters

Article Language

Species

Sex

Age

Other

Search Results

12 results

Results by year