Rajan Giri - Search Results

Year	Number of Results
2008	1
2009	1
2010	3
2012	1
2020	2
2021	1
2022	1
2023	1
2026	0

1

Further studies on C2'-substituted 1-phenylbenzazepines as dopamine D1 receptor ligands.

Giri R, Namballa HK, Sarker A, Alberts I, Harding WW. Giri R, et al. Bioorg Chem. 2022 Oct;127:105953. doi: 10.1016/j.bioorg.2022.105953. Epub 2022 Jun 22. Bioorg Chem. 2022. PMID: 35772367

2

Synthesis and dopamine receptor pharmacological evaluations on ring C ortho halogenated 1-phenylbenzazepines.

Giri R, Namballa HK, Sarker A, Alberts I, Harding WW. Giri R, et al. Bioorg Med Chem Lett. 2020 Aug 15;30(16):127305. doi: 10.1016/j.bmcl.2020.127305. Epub 2020 Jun 4. Bioorg Med Chem Lett. 2020. PMID: 32631525 Free PMC article.

3

Structure-Activity Relationship Studies on 6-Chloro-1-phenylbenzazepines Leads to the Identification of a New Dopamine D1 Receptor Antagonist.

Giri R, Namballa HK, Emogaje V, Harding WW. Giri R, et al. Molecules. 2023 Aug 11;28(16):6010. doi: 10.3390/molecules28166010. Molecules. 2023. PMID: 37630262 Free PMC article.

4

Synthesis, pharmacological evaluations, and molecular docking studies on a new 1,3,4,11b-tetrahydro-1H-fluoreno[9,1-cd]azepine framework: Rigidification of D₁ receptor selective 1-phenylbenzazepines and discovery of a new 5-HT₆ receptor scaffold.

Giri R, Alberts I, Harding WW. Giri R, et al. Chem Biol Drug Des. 2020 Aug;96(2):825-835. doi: 10.1111/cbdd.13691. Epub 2020 Apr 22. Chem Biol Drug Des. 2020. PMID: 32279445 Free PMC article.

5

Novel theranostic agent for PET imaging and targeted radiopharmaceutical therapy of tumour-infiltrating immune cells in glioma.

Foster A, Nigam S, Tatum DS, Raphael I, Xu J, Kumar R, Plakseychuk E, Latoche JD, Vincze S, Li B, Giri R, McCarl LH, Edinger R, Ak M, Peddagangireddy V, Foley LM, Hitchens TK, Colen RR, Pollack IF, Panigrahy A, Magda D, Anderson CJ, Edwards WB, Kohanbash G. Foster A, et al. Among authors: giri r. EBioMedicine. 2021 Sep;71:103571. doi: 10.1016/j.ebiom.2021.103571. Epub 2021 Sep 13. EBioMedicine. 2021. PMID: 34530385 Free PMC article.

6

9-Amino acridine pharmacokinetics, brain distribution, and in vitro/in vivo efficacy against malignant glioma.

Teitelbaum AM, Gallardo JL, Bedi J, Giri R, Benoit AR, Olin MR, Morizio KM, Ohlfest JR, Remmel RP, Ferguson DM. Teitelbaum AM, et al. Among authors: giri r. Cancer Chemother Pharmacol. 2012 Jun;69(6):1519-27. doi: 10.1007/s00280-012-1855-5. Epub 2012 Mar 9. Cancer Chemother Pharmacol. 2012. PMID: 22402637

7

Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-kappaB and AP-1 mediated transcriptional activation: Their possible utilization as anti-inflammatory and anti-cancer agents.

Giri RS, Thaker HM, Giordano T, Williams J, Rogers D, Vasu KK, Sudarsanam V. Giri RS, et al. Bioorg Med Chem. 2010 Apr 1;18(7):2796-808. doi: 10.1016/j.bmc.2010.01.007. Epub 2010 Jan 11. Bioorg Med Chem. 2010. PMID: 20335039

8

Synthesis and evaluation of quinazolinone derivatives as inhibitors of NF-kappaB, AP-1 mediated transcription and eIF-4E mediated translational activation: inhibitors of multi-pathways involve in cancer.

Giri RS, Thaker HM, Giordano T, Chen B, Nuthalapaty S, Vasu KK, Sudarsanam V. Giri RS, et al. Eur J Med Chem. 2010 Sep;45(9):3558-63. doi: 10.1016/j.ejmech.2010.04.038. Epub 2010 May 7. Eur J Med Chem. 2010. PMID: 20557982

9

Synthesis and cancer cell cytotoxicity of substituted xanthenes.

Giri R, Goodell JR, Xing C, Benoit A, Kaur H, Hiasa H, Ferguson DM. Giri R, et al. Bioorg Med Chem. 2010 Feb 15;18(4):1456-63. doi: 10.1016/j.bmc.2010.01.018. Epub 2010 Jan 11. Bioorg Med Chem. 2010. PMID: 20129790

10

Design, synthesis and characterization of novel 2-(2,4-disubstituted-thiazole-5-yl)-3-aryl-3H-quinazoline-4-one derivatives as inhibitors of NF-kappaB and AP-1 mediated transcription activation and as potential anti-inflammatory agents.

Giri RS, Thaker HM, Giordano T, Williams J, Rogers D, Sudersanam V, Vasu KK. Giri RS, et al. Eur J Med Chem. 2009 May;44(5):2184-9. doi: 10.1016/j.ejmech.2008.10.031. Epub 2008 Nov 5. Eur J Med Chem. 2009. PMID: 19064304

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