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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
2002 1
2004 2
2005 3
2006 5
2007 8
2008 5
2009 4
2010 1
2011 2
2012 3
2013 4
2014 5
2015 7
2016 5
2017 5
2018 4
2019 1
2020 2
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63 results
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Page 1
Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants.
Marek M, Shaik TB, Heimburg T, Chakrabarti A, Lancelot J, Ramos-Morales E, Da Veiga C, Kalinin D, Melesina J, Robaa D, Schmidtkunz K, Suzuki T, Holl R, Ennifar E, Pierce RJ, Jung M, Sippl W, Romier C. Marek M, et al. Among authors: pierce rj. J Med Chem. 2018 Nov 21;61(22):10000-10016. doi: 10.1021/acs.jmedchem.8b01087. Epub 2018 Nov 8. J Med Chem. 2018. PMID: 30347148
Structure-Reactivity Relationships on Substrates and Inhibitors of the Lysine Deacylase Sirtuin 2 from Schistosoma mansoni (SmSirt2).
Monaldi D, Rotili D, Lancelot J, Marek M, Wössner N, Lucidi A, Tomaselli D, Ramos-Morales E, Romier C, Pierce RJ, Mai A, Jung M. Monaldi D, et al. Among authors: pierce rj. J Med Chem. 2019 Oct 10;62(19):8733-8759. doi: 10.1021/acs.jmedchem.9b00638. Epub 2019 Sep 20. J Med Chem. 2019. PMID: 31496251
Combattre les maladies négligées en ciblant sélectivement leurs enzymes épigénétiques : le cas de la désacétylase 8 (HDAC8) de Schistosoma mansoni.
Marek M, Shaik TB, Jung M, Sippl W, Pierce RJ, Romier C. Marek M, et al. Among authors: pierce rj. Biol Aujourdhui. 2016;210(4):311-320. doi: 10.1051/jbio/2017001. Epub 2017 Mar 22. Biol Aujourdhui. 2016. PMID: 28327287 French.
Schistosome sirtuins as drug targets.
Lancelot J, Cabezas-Cruz A, Caby S, Marek M, Schultz J, Romier C, Sippl W, Jung M, Pierce RJ. Lancelot J, et al. Among authors: pierce rj. Future Med Chem. 2015;7(6):765-82. doi: 10.4155/fmc.15.24. Future Med Chem. 2015. PMID: 25996069 Free article. Review.
HDAC8: a multifaceted target for therapeutic interventions.
Chakrabarti A, Oehme I, Witt O, Oliveira G, Sippl W, Romier C, Pierce RJ, Jung M. Chakrabarti A, et al. Among authors: pierce rj. Trends Pharmacol Sci. 2015 Jul;36(7):481-92. doi: 10.1016/j.tips.2015.04.013. Epub 2015 May 23. Trends Pharmacol Sci. 2015. PMID: 26013035 Free article. Review.
Drugging the schistosome zinc-dependent HDACs: current progress and future perspectives.
Marek M, Oliveira G, Pierce RJ, Jung M, Sippl W, Romier C. Marek M, et al. Among authors: pierce rj. Future Med Chem. 2015;7(6):783-800. doi: 10.4155/fmc.15.25. Future Med Chem. 2015. PMID: 25996070 Free article. Review.
How has the genomics era impacted schistosomiasis drug discovery?
Oliveira G, Pierce RJ. Oliveira G, et al. Among authors: pierce rj. Future Med Chem. 2015;7(6):685-7. doi: 10.4155/fmc.15.30. Future Med Chem. 2015. PMID: 25996060 Free article. No abstract available.
Epigenetic control of gene function in schistosomes: a source of therapeutic targets?
Cabezas-Cruz A, Lancelot J, Caby S, Oliveira G, Pierce RJ. Cabezas-Cruz A, et al. Among authors: pierce rj. Front Genet. 2014 Sep 10;5:317. doi: 10.3389/fgene.2014.00317. eCollection 2014. Front Genet. 2014. PMID: 25309576 Free PMC article. Review.
Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as SmHDAC8 Inhibitors for the Treatment of Schistosomiasis.
Bayer T, Chakrabarti A, Lancelot J, Shaik TB, Hausmann K, Melesina J, Schmidtkunz K, Marek M, Erdmann F, Schmidt M, Robaa D, Romier C, Pierce RJ, Jung M, Sippl W. Bayer T, et al. Among authors: pierce rj. ChemMedChem. 2018 Aug 10;13(15):1517-1529. doi: 10.1002/cmdc.201800238. Epub 2018 Jul 4. ChemMedChem. 2018. PMID: 29806110
A Novel Class of Schistosoma mansoni Histone Deacetylase 8 (HDAC8) Inhibitors Identified by Structure-Based Virtual Screening and In Vitro Testing.
Simoben CV, Robaa D, Chakrabarti A, Schmidtkunz K, Marek M, Lancelot J, Kannan S, Melesina J, Shaik TB, Pierce RJ, Romier C, Jung M, Sippl W. Simoben CV, et al. Among authors: pierce rj. Molecules. 2018 Mar 2;23(3):566. doi: 10.3390/molecules23030566. Molecules. 2018. PMID: 29498707 Free PMC article.
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