Transient Competitive Inhibition Bypasses the Binding Site Barrier to Improve Tumor Penetration of Trastuzumab and Enhance T-DM1 Efficacy.
Cancer Res. 2021 Aug 1;81(15):4145-4154. doi: 10.1158/0008-5472.CAN-20-3822. Epub 2021 Mar 16.
Cancer Res. 2021.
PMID: 33727230
Free PMC article.