Haaksma E[au] - Search Results

Year	Number of Results
1987	1
1989	1
1990	1
1991	1
1992	1
2000	4
2003	1
2005	1
2008	4
2009	3
2010	1
2012	3
2013	3
2015	2
2022	1
2023	0

1

Histamine receptors: subclasses and specific ligands.

Haaksma EE, Leurs R, Timmerman H. Haaksma EE, et al. Pharmacol Ther. 1990;47(1):73-104. doi: 10.1016/0163-7258(90)90046-5. Pharmacol Ther. 1990. PMID: 2195558 Review.

2

Predicting ligand interactions with ABC transporters in ADME.

Demel MA, Krämer O, Ettmayer P, Haaksma EE, Ecker GF. Demel MA, et al. Among authors: haaksma ee. Chem Biodivers. 2009 Nov;6(11):1960-9. doi: 10.1002/cbdv.200900138. Chem Biodivers. 2009. PMID: 19937827 Review.

3

opnMe.com: a digital initiative for sharing tools with the biomedical research community.

Gollner A, Köster M, Nicklin P, Trieselmann T, Klein E, Vlach J, Heine C, Grundl M, Ramharter J, Wyatt D, Chaturvedi M, Ciulli A, Carter KC, Müller S, Bischoff D, Ettmayer P, Haaksma E, Mack J, McConnell D, Stenkamp D, Weinstabl H, Zentgraf M, Wood CR, Montel F. Gollner A, et al. Among authors: haaksma e. Nat Rev Drug Discov. 2022 Jul;21(7):475-476. doi: 10.1038/d41573-022-00071-9. Nat Rev Drug Discov. 2022. PMID: 35459938 No abstract available.

4

In silico prediction of substrate properties for ABC-multidrug transporters.

Demel MA, Schwaha R, Krämer O, Ettmayer P, Haaksma EE, Ecker GF. Demel MA, et al. Among authors: haaksma ee. Expert Opin Drug Metab Toxicol. 2008 Sep;4(9):1167-80. doi: 10.1517/17425255.4.9.1167. Expert Opin Drug Metab Toxicol. 2008. PMID: 18721111 Review.

5

A new generation of anti-histamines: Histamine H4 receptor antagonists on their way to the clinic.

Engelhardt H, Smits RA, Leurs R, Haaksma E, de Esch IJ. Engelhardt H, et al. Among authors: haaksma e. Curr Opin Drug Discov Devel. 2009 Sep;12(5):628-43. Curr Opin Drug Discov Devel. 2009. PMID: 19736622 Review.

6

Detailed structure-activity relationship of indolecarboxamides as H4 receptor ligands.

Engelhardt H, de Esch IJ, Kuhn D, Smits RA, Zuiderveld OP, Dobler J, Mayer M, Lips S, Arnhof H, Scharn D, Haaksma EE, Leurs R. Engelhardt H, et al. Among authors: haaksma ee. Eur J Med Chem. 2012 Aug;54:660-8. doi: 10.1016/j.ejmech.2012.06.016. Epub 2012 Jun 18. Eur J Med Chem. 2012. PMID: 22749391

7

Combining quantum mechanical ligand conformation analysis and protein modeling to elucidate GPCR-ligand binding modes.

Schultes S, Engelhardt H, Roumen L, Zuiderveld OP, Haaksma EE, de Esch IJ, Leurs R, de Graaf C. Schultes S, et al. Among authors: haaksma ee. ChemMedChem. 2013 Jan;8(1):49-53. doi: 10.1002/cmdc.201200412. Epub 2012 Nov 19. ChemMedChem. 2013. PMID: 23161844

8

Linking agonist binding to histamine H1 receptor activation.

Jongejan A, Bruysters M, Ballesteros JA, Haaksma E, Bakker RA, Pardo L, Leurs R. Jongejan A, et al. Among authors: haaksma e. Nat Chem Biol. 2005 Jul;1(2):98-103. doi: 10.1038/nchembio714. Epub 2005 Jun 19. Nat Chem Biol. 2005. PMID: 16408006

9

Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach.

Smits RA, de Esch IJ, Zuiderveld OP, Broeker J, Sansuk K, Guaita E, Coruzzi G, Adami M, Haaksma E, Leurs R. Smits RA, et al. Among authors: haaksma e. J Med Chem. 2008 Dec 25;51(24):7855-65. doi: 10.1021/jm800876b. J Med Chem. 2008. PMID: 19053770

10

Heterocyclic thrombin inhibitors. Part 1: design and synthesis of amidino-phenoxy quinoline derivatives.

Ries UJ, Priepke HW, Hauel NH, Haaksma EE, Stassen JM, Wienen W, Nar H. Ries UJ, et al. Among authors: haaksma ee. Bioorg Med Chem Lett. 2003 Jul 21;13(14):2291-5. doi: 10.1016/s0960-894x(03)00442-6. Bioorg Med Chem Lett. 2003. PMID: 12824020

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