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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
1974 1
1975 1
1976 1
1977 2
1978 1
1980 8
1981 4
1982 6
1983 1
1984 4
1985 4
1987 4
1988 3
1989 3
1990 4
1991 2
1992 2
1993 1
1994 1
1995 6
1996 3
1997 4
1998 2
1999 4
2000 3
2001 8
2002 7
2003 5
2004 4
2005 5
2006 8
2007 6
2008 9
2009 7
2010 11
2011 7
2012 6
2013 11
2014 8
2015 9
2016 11
2017 13
2018 5
2019 12
2020 6
2021 2
2022 2
2023 2
2024 4

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225 results

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Page 1
Allosteric ligands for the pharmacologically dark receptors GPR68 and GPR65.
Huang XP, Karpiak J, Kroeze WK, Zhu H, Chen X, Moy SS, Saddoris KA, Nikolova VD, Farrell MS, Wang S, Mangano TJ, Deshpande DA, Jiang A, Penn RB, Jin J, Koller BH, Kenakin T, Shoichet BK, Roth BL. Huang XP, et al. Among authors: kenakin t. Nature. 2015 Nov 26;527(7579):477-83. doi: 10.1038/nature15699. Epub 2015 Nov 9. Nature. 2015. PMID: 26550826 Free PMC article.
Editors in Chief Overview.
Trist DG, Kenakin TP. Trist DG, et al. Among authors: kenakin tp. Curr Opin Pharmacol. 2017 Aug;35:iv-v. doi: 10.1016/j.coph.2017.11.003. Curr Opin Pharmacol. 2017. PMID: 29241830 No abstract available.
Community guidelines for GPCR ligand bias: IUPHAR review 32.
Kolb P, Kenakin T, Alexander SPH, Bermudez M, Bohn LM, Breinholt CS, Bouvier M, Hill SJ, Kostenis E, Martemyanov KA, Neubig RR, Onaran HO, Rajagopal S, Roth BL, Selent J, Shukla AK, Sommer ME, Gloriam DE. Kolb P, et al. Among authors: kenakin t. Br J Pharmacol. 2022 Jul;179(14):3651-3674. doi: 10.1111/bph.15811. Epub 2022 Mar 27. Br J Pharmacol. 2022. PMID: 35106752 Free PMC article. Review.
Biased agonism.
Kenakin T. Kenakin T. F1000 Biol Rep. 2009 Nov 26;1:87. doi: 10.3410/B1-87. F1000 Biol Rep. 2009. PMID: 20948603 Free PMC article.
Bias translation: The final frontier?
Kenakin T. Kenakin T. Br J Pharmacol. 2024 May;181(9):1345-1360. doi: 10.1111/bph.16335. Epub 2024 Feb 29. Br J Pharmacol. 2024. PMID: 38424747 Review.
Receptor theory.
Kenakin T. Kenakin T. Curr Protoc Pharmacol. 2008 Jun;Chapter 1:Unit1.2. doi: 10.1002/0471141755.ph0102s41. Curr Protoc Pharmacol. 2008. PMID: 22294216
Signaling bias in drug discovery.
Kenakin T. Kenakin T. Expert Opin Drug Discov. 2017 Apr;12(4):321-333. doi: 10.1080/17460441.2017.1297417. Epub 2017 Mar 9. Expert Opin Drug Discov. 2017. PMID: 28277840 Review.
225 results