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Diltiazem inhibition of cytochrome P-450 3A activity is due to metabolite intermediate complex formation.
J Pharmacol Exp Ther. 1999 Sep;290(3):1116-25.
J Pharmacol Exp Ther. 1999.
PMID: 10454485
An in vitro model for predicting in vivo inhibition of cytochrome P450 3A4 by metabolic intermediate complex formation.
Mayhew BS, Jones DR, Hall SD.
Mayhew BS, et al.
Drug Metab Dispos. 2000 Sep;28(9):1031-7.
Drug Metab Dispos. 2000.
PMID: 10950845
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