Schaffhauser H[au] - Search Results

Year	Number of Results
1997	3
1998	5
1999	1
2000	1
2001	1
2002	1
2003	4
2004	8
2005	5
2006	1
2007	2
2008	4
2009	3
2010	1
2011	3
2012	3
2017	1
2022	1
2023	0

1

5-HT6 receptor antagonists as potential therapeutics for cognitive impairment.

Rossé G, Schaffhauser H. Rossé G, et al. Among authors: schaffhauser h. Curr Top Med Chem. 2010;10(2):207-21. doi: 10.2174/156802610790411036. Curr Top Med Chem. 2010. PMID: 20166958 Review.

2

Detection of low level histamine H3 receptor occupancy by autoradiography.

Le S, Finn JP, Larijani ME, Marino MJ, Schaffhauser H. Le S, et al. Among authors: schaffhauser h. J Neurosci Methods. 2009 Dec 15;185(1):70-5. doi: 10.1016/j.jneumeth.2009.09.015. Epub 2009 Sep 16. J Neurosci Methods. 2009. PMID: 19765611

3

Metabotropic glutamate receptors: potential drug targets for the treatment of schizophrenia.

Chavez-Noriega LE, Schaffhauser H, Campbell UC. Chavez-Noriega LE, et al. Among authors: schaffhauser h. Curr Drug Targets CNS Neurol Disord. 2002 Jun;1(3):261-81. doi: 10.2174/1568007023339337. Curr Drug Targets CNS Neurol Disord. 2002. PMID: 12769619 Review.

4

A high quality, industrial data set for binding affinity prediction: performance comparison in different early drug discovery scenarios.

Tosstorff A, Rudolph MG, Cole JC, Reutlinger M, Kramer C, Schaffhauser H, Nilly A, Flohr A, Kuhn B. Tosstorff A, et al. Among authors: schaffhauser h. J Comput Aided Mol Des. 2022 Oct;36(10):753-765. doi: 10.1007/s10822-022-00478-x. Epub 2022 Sep 25. J Comput Aided Mol Des. 2022. PMID: 36153472

5

Novel brain penetrant benzofuropiperidine 5-HT₆ receptor antagonists.

Sundar BG, Bailey TR, Dunn DD, Bacon ER, Salvino JM, Morton GC, Aimone LD, Zeqi H, Mathiasen JR, Dicamillo A, Huffman MJ, McKenna BA, Kopec K, Lu LD, Brown R, Qian J, Angeles T, Connors T, Spais C, Holskin B, Galinis D, Duzic E, Schaffhauser H, Rosse GC. Sundar BG, et al. Among authors: schaffhauser h. Bioorg Med Chem Lett. 2012 Jan 1;22(1):120-3. doi: 10.1016/j.bmcl.2011.11.050. Epub 2011 Nov 22. Bioorg Med Chem Lett. 2012. PMID: 22153937

6

Discovery of the first low-shift positive allosteric modulators for the muscarinic M1 receptor.

Flohr A, Hutter R, Mueller B, Bohnert C, Pellisson M, Schaffhauser H. Flohr A, et al. Among authors: schaffhauser h. Bioorg Med Chem Lett. 2017 Dec 15;27(24):5415-5419. doi: 10.1016/j.bmcl.2017.11.008. Epub 2017 Nov 6. Bioorg Med Chem Lett. 2017. PMID: 29146472

7

Dimebolin is a 5-HT6 antagonist with acute cognition enhancing activities.

Schaffhauser H, Mathiasen JR, Dicamillo A, Huffman MJ, Lu LD, McKenna BA, Qian J, Marino MJ. Schaffhauser H, et al. Biochem Pharmacol. 2009 Oct 15;78(8):1035-42. doi: 10.1016/j.bcp.2009.06.021. Epub 2009 Jun 21. Biochem Pharmacol. 2009. PMID: 19549510

8

Challenges in the development of mGluR5 positive allosteric modulators: the discovery of CPPHA.

Zhao Z, Wisnoski DD, O'Brien JA, Lemaire W, Williams DL Jr, Jacobson MA, Wittman M, Ha SN, Schaffhauser H, Sur C, Pettibone DJ, Duggan ME, Conn PJ, Hartman GD, Lindsley CW. Zhao Z, et al. Among authors: schaffhauser h. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1386-91. doi: 10.1016/j.bmcl.2006.11.081. Epub 2006 Dec 3. Bioorg Med Chem Lett. 2007. PMID: 17210250

9

Biphenyl-indanones: allosteric potentiators of the metabotropic glutamate subtype 2 receptor.

Bonnefous C, Vernier JM, Hutchinson JH, Gardner MF, Cramer M, James JK, Rowe BA, Daggett LP, Schaffhauser H, Kamenecka TM. Bonnefous C, et al. Among authors: schaffhauser h. Bioorg Med Chem Lett. 2005 Oct 1;15(19):4354-8. doi: 10.1016/j.bmcl.2005.06.062. Bioorg Med Chem Lett. 2005. PMID: 16046122

10

Phenyl-tetrazolyl acetophenones: discovery of positive allosteric potentiatiors for the metabotropic glutamate 2 receptor.

Pinkerton AB, Vernier JM, Schaffhauser H, Rowe BA, Campbell UC, Rodriguez DE, Lorrain DS, Baccei CS, Daggett LP, Bristow LJ. Pinkerton AB, et al. Among authors: schaffhauser h. J Med Chem. 2004 Aug 26;47(18):4595-9. doi: 10.1021/jm040088h. J Med Chem. 2004. PMID: 15317469

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