Similar articles for PMID: 12215417

Year	Number of Results
1989	1
1993	1
1995	2
1996	2
1997	3
1998	7
1999	4
2000	8
2001	7
2002	14
2003	14
2004	10
2005	17
2006	10
2007	11
2008	18
2009	13
2010	12
2011	17
2012	8
2013	13
2014	12
2015	2
2016	7
2017	7
2018	5
2019	12
2020	2
2021	5
2022	3
2023	3
2024	0

1

Structural basis for AMPA receptor activation and ligand selectivity: crystal structures of five agonist complexes with the GluR2 ligand-binding core.

Hogner A, Kastrup JS, Jin R, Liljefors T, Mayer ML, Egebjerg J, Larsen IK, Gouaux E. Hogner A, et al. J Mol Biol. 2002 Sep 6;322(1):93-109. doi: 10.1016/s0022-2836(02)00650-2. J Mol Biol. 2002. PMID: 12215417

2

Tyr702 is an important determinant of agonist binding and domain closure of the ligand-binding core of GluR2.

Frandsen A, Pickering DS, Vestergaard B, Kasper C, Nielsen BB, Greenwood JR, Campiani G, Fattorusso C, Gajhede M, Schousboe A, Kastrup JS. Frandsen A, et al. Mol Pharmacol. 2005 Mar;67(3):703-13. doi: 10.1124/mol.104.002931. Epub 2004 Dec 9. Mol Pharmacol. 2005. PMID: 15591246

3

Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H- tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist.

Vogensen SB, Jensen HS, Stensbøl TB, Frydenvang K, Bang-Andersen B, Johansen TN, Egebjerg J, Krogsgaard-Larsen P. Vogensen SB, et al. Chirality. 2000 Nov;12(10):705-13. doi: 10.1002/1520-636X(2000)12:10<705::AID-CHIR2>3.0.CO;2-9. Chirality. 2000. PMID: 11054828

4

Structural determinants of agonist-specific kinetics at the ionotropic glutamate receptor 2.

Holm MM, Lunn ML, Traynelis SF, Kastrup JS, Egebjerg J. Holm MM, et al. Proc Natl Acad Sci U S A. 2005 Aug 23;102(34):12053-8. doi: 10.1073/pnas.0505522102. Epub 2005 Aug 11. Proc Natl Acad Sci U S A. 2005. PMID: 16099829 Free PMC article.

5

A binding site tyrosine shapes desensitization kinetics and agonist potency at GluR2. A mutagenic, kinetic, and crystallographic study.

Holm MM, Naur P, Vestergaard B, Geballe MT, Gajhede M, Kastrup JS, Traynelis SF, Egebjerg J. Holm MM, et al. J Biol Chem. 2005 Oct 21;280(42):35469-76. doi: 10.1074/jbc.M507800200. Epub 2005 Aug 15. J Biol Chem. 2005. PMID: 16103115 Free article.

6

Mechanism of activation and selectivity in a ligand-gated ion channel: structural and functional studies of GluR2 and quisqualate.

Jin R, Horning M, Mayer ML, Gouaux E. Jin R, et al. Biochemistry. 2002 Dec 31;41(52):15635-43. doi: 10.1021/bi020583k. Biochemistry. 2002. PMID: 12501192

7

Excitatory amino acid receptor ligands: resolution, absolute stereochemistry, and enantiopharmacology of 2-amino-3-(4-butyl-3-hydroxyisoxazol-5-yl)propionic acid.

Johansen TN, Ebert B, Bräuner-Osborne H, Didriksen M, Christensen IT, Søby KK, Madsen U, Krogsgaard-Larsen P, Brehm L. Johansen TN, et al. J Med Chem. 1998 Mar 12;41(6):930-9. doi: 10.1021/jm9706731. J Med Chem. 1998. PMID: 9526567

8

Structures of the ligand-binding core of iGluR2 in complex with the agonists (R)- and (S)-2-amino-3-(4-hydroxy-1,2,5-thiadiazol-3-yl)propionic acid explain their unusual equipotency.

Beich-Frandsen M, Pickering DS, Mirza O, Johansen TN, Greenwood J, Vestergaard B, Schousboe A, Gajhede M, Liljefors T, Kastrup JS. Beich-Frandsen M, et al. J Med Chem. 2008 Mar 13;51(5):1459-63. doi: 10.1021/jm701126w. Epub 2008 Feb 13. J Med Chem. 2008. PMID: 18269227

9

Three-dimensional structure of the ligand-binding core of GluR2 in complex with the agonist (S)-ATPA: implications for receptor subunit selectivity.

Lunn ML, Hogner A, Stensbøl TB, Gouaux E, Egebjerg J, Kastrup JS. Lunn ML, et al. J Med Chem. 2003 Feb 27;46(5):872-5. doi: 10.1021/jm021020+. J Med Chem. 2003. PMID: 12593667

10

Tuning activation of the AMPA-sensitive GluR2 ion channel by genetic adjustment of agonist-induced conformational changes.

Armstrong N, Mayer M, Gouaux E. Armstrong N, et al. Proc Natl Acad Sci U S A. 2003 May 13;100(10):5736-41. doi: 10.1073/pnas.1037393100. Epub 2003 May 2. Proc Natl Acad Sci U S A. 2003. PMID: 12730367 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

229 results

Results by year