Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.
Varga BR, Uprety R, Paul B, Knoll A, Ramos-Gonzalez N, Appourchaux K, Taylor T, Turgutalp B, Shinouchi R, Eans SO, Williams AK, Vasquez-Grinnell SG, Zaidi S, Nazarova AL, Varadi A, Le Rouzic V, Brown TG, Martinez S, Ansonoff M, Dardashti RN, Hunkele A, Subrath J, Welch M, Xu J, Rossi GC, Pintar J, Pasternak GW, Katritch V, McLaughlin JP, Pan YX, Majumdar S.
Varga BR, et al.
ACS Chem Neurosci. 2025 Jul 16;16(14):2714-2737. doi: 10.1021/acschemneuro.5c00312. Epub 2025 Jun 26.
ACS Chem Neurosci. 2025.
PMID: 40566691