Discovery of Naphthyridinone Derivatives as Selective and Potent PKMYT1 Inhibitors with Antitumor Efficacy.
Chen B, Liu X, Mu T, Xu J, Zhao D, Dey F, Tang Y, Xu Z, Yang J, Huang K, Li C, Chen S, Zhu S, Wang S, Yao X, Yan Z, Tu Y, Dai Y, Qiu H, Yang J, Jiang T, Qi Y, Li Y, Shen HC, Zhu W, Tan X, Wu J.
Chen B, et al. Among authors: yan z.
J Med Chem. 2025 Apr 24;68(8):8497-8515. doi: 10.1021/acs.jmedchem.5c00114. Epub 2025 Apr 8.
J Med Chem. 2025.
PMID: 40198752