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Quoted phrase not found in phrase index: "benzopseudoxazole"
Page 1
Zonisamide.
Kadian R, Patel P, Kumar A. Kadian R, et al. 2025 Feb 15. In: StatPearls [Internet]. Treasure Island (FL): StatPearls Publishing; 2026 Jan–. 2025 Feb 15. In: StatPearls [Internet]. Treasure Island (FL): StatPearls Publishing; 2026 Jan–. PMID: 29939680 Free Books & Documents.
Zonisamide is a sulfonamide antiepileptic drug that is chemically distinct from other antiepileptic medications. As a 1,2-benzisoxazole derivative, it may be indicated for both epileptic and non-epileptic conditions. ...
Zonisamide is a sulfonamide antiepileptic drug that is chemically distinct from other antiepileptic medications. As a 1,2-b …
Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer.
Sharma S, Chung CY, Uryu S, Petrovic J, Cao J, Rickard A, Nady N, Greasley S, Johnson E, Brodsky O, Khan S, Wang H, Wang Z, Zhang Y, Tsaparikos K, Chen L, Mazurek A, Lapek J, Kung PP, Sutton S, Richardson PF, Greenwald EC, Yamazaki S, Jones R, Maegley KA, Bingham P, Lam H, Stupple AE, Kamal A, Chueh A, Cuzzupe A, Morrow BJ, Ren B, Carrasco-Pozo C, Tan CW, Bhuva DD, Allan E, Surgenor E, Vaillant F, Pehlivanoglu H, Falk H, Whittle JR, Newman J, Cursons J, Doherty JP, White KL, MacPherson L, Devlin M, Dennis ML, Hattarki MK, De Silva M, Camerino MA, Butler MS, Dolezal O, Pilling P, Foitzik R, Stupple PA, Lagiakos HR, Walker SR, Hediyeh-Zadeh S, Nuttall S, Spall SK, Charman SA, Connor T, Peat TS, Avery VM, Bozikis YE, Yang Y, Zhang M, Monahan BJ, Voss AK, Thomas T, Street IP, Dawson SJ, Dawson MA, Lindeman GJ, Davis MJ, Visvader JE, Paul TA. Sharma S, et al. Cell Chem Biol. 2023 Oct 19;30(10):1191-1210.e20. doi: 10.1016/j.chembiol.2023.07.005. Epub 2023 Aug 8. Cell Chem Biol. 2023. PMID: 37557181 Free article.
Here we describe identification of a highly potent, selective, and orally bioavailable KAT6A/KAT6B inhibitor CTx-648 (PF-9363), derived from a benzisoxazole series, which demonstrates anti-tumor activity in correlation with H3K23Ac inhibition in KAT6A over-expressing breas …
Here we describe identification of a highly potent, selective, and orally bioavailable KAT6A/KAT6B inhibitor CTx-648 (PF-9363), derived from …
Aripiprazole.
Ardiana F, Lestari ML, Indrayanto G. Ardiana F, et al. Profiles Drug Subst Excip Relat Methodol. 2013;38:35-85. doi: 10.1016/B978-0-12-407691-4.00002-2. Profiles Drug Subst Excip Relat Methodol. 2013. PMID: 23668402 Review.
Aripiprazole is an atypical antipsychotic drug which belongs to the benzisoxazole derivatives. Aripiprazole is available in many salts and polymorphs forms. X-ray diffraction, IR spectroscopy, and DSC could be used for differentiating the polymorphs of aripiprazole. ...
Aripiprazole is an atypical antipsychotic drug which belongs to the benzisoxazole derivatives. Aripiprazole is available in many salt …
Risperidone.
Cohen LJ. Cohen LJ. Pharmacotherapy. 1994 May-Jun;14(3):253-65. Pharmacotherapy. 1994. PMID: 7524043 Review.
Risperidone, a benzisoxazole derivative, is a novel antipsychotic agent that has an extremely strong binding affinity for serotonin 5-HT2 receptors, a strong binding affinity for dopamine D2 receptors, and a high affinity for alpha 1- and alpha 2-adrenergic receptors and h …
Risperidone, a benzisoxazole derivative, is a novel antipsychotic agent that has an extremely strong binding affinity for serotonin 5 …
3-{[5-(4-Bromo-phen-yl)imidazo[2,1-b][1,3,4]thia-diazol-2-yl]meth-yl}-1,2-benzoxazole.
Banu A, Ziaulla M, Begum NS, Lamani RS, Khazi IM. Banu A, et al. Acta Crystallogr Sect E Struct Rep Online. 2010 Dec 18;67(Pt 1):o154. doi: 10.1107/S1600536810052232. Acta Crystallogr Sect E Struct Rep Online. 2010. PMID: 21522661 Free PMC article.
In the title compound, C(18)H(11)BrN(4)OS, the imidazothia-diazole and benzisoxazole rings are individually planar with maximum deviations of 0.025 (3) 0.015 (4) A, respectively, and are inclined at an angle of 23.51 (7) with respect to each other. ...
In the title compound, C(18)H(11)BrN(4)OS, the imidazothia-diazole and benzisoxazole rings are individually planar with maximum devia …
3-{[6-(4-Chloro-phen-yl)imidazo[2,1-b][1,3,4]thia-diazol-2-yl]meth-yl}-1,2-benzoxazole.
Banu A, Ziaulla M, Begum NS, Lamani RS, Khazi IM. Banu A, et al. Acta Crystallogr Sect E Struct Rep Online. 2011 Feb 12;67(Pt 3):o617-8. doi: 10.1107/S1600536811004582. Acta Crystallogr Sect E Struct Rep Online. 2011. PMID: 21522374 Free PMC article.
In the title compound, C(18)H(11)ClN(4)OS, the benzisoxazole and imidazothia-diazole rings are inclined at an angle of 23.81 (7) with respect to each other. ...
In the title compound, C(18)H(11)ClN(4)OS, the benzisoxazole and imidazothia-diazole rings are inclined at an angle of 23.81 (7) wit …
1,2-Benzisoxazole compounds: a patent review (2009 - 2014).
Uto Y. Uto Y. Expert Opin Ther Pat. 2015 Jun;25(6):643-62. doi: 10.1517/13543776.2015.1027192. Epub 2015 Mar 23. Expert Opin Ther Pat. 2015. PMID: 25800253 Review.
AREAS COVERED: This review puts emphasis on the recent progress in therapeutically attractive benzisoxazole derivatives especially 1,2-benzisoxazoles, which were published in the patent literature between 2009 and 2014. ...This review also covers the examples of benziso …
AREAS COVERED: This review puts emphasis on the recent progress in therapeutically attractive benzisoxazole derivatives especially 1, …
Monoamine oxidase inhibition properties of 2,1-benzisoxazole derivatives.
Shetnev A, Kotov A, Kunichkina A, Proskurina I, Baykov S, Korsakov M, Petzer A, Petzer JP. Shetnev A, et al. Mol Divers. 2024 Jun;28(3):1009-1021. doi: 10.1007/s11030-023-10628-4. Epub 2023 Mar 19. Mol Divers. 2024. PMID: 36934384 Free PMC article.
It is interesting to note that 3-(2-aminoethoxy)-1,2-benzisoxazole derivatives, the 1,2-benzisoxazole, zonisamide, as well as the isoxazole compound, leflunomide, have been described as MAO inhibitors. This is however the first report of …
It is interesting to note that 3-(2-aminoethoxy)-1,2-benzisoxazole derivatives, the 1,2-benzisoxazole …
Novel and efficient synthesis of 5-chloro-6-methoxy-3-(2-((1-(aryl)-1H-1,2,3-triazol-4-yl)methoxy)ethyl)benzo[d]isoxazole derivatives as new α-glucosidase inhibitors.
Mudireddy RR, Gundla R, Koraboina CP, Velavalapalli VM, Sarma Dhulipalla VV, Burle GS, Jonnalagadda SB, Katari NK. Mudireddy RR, et al. Biochem Biophys Rep. 2025 Jun 5;43:102074. doi: 10.1016/j.bbrep.2025.102074. eCollection 2025 Sep. Biochem Biophys Rep. 2025. PMID: 40546344 Free PMC article.
A new series of benzisoxazole derivatives (9a-o) were designed by using molecular hybridization approach and synthesized via click-chemistry. ...
A new series of benzisoxazole derivatives (9a-o) were designed by using molecular hybridization approach and synthesized via click-ch …
3-Benzyl-5-methyl-1,2-benzoxazole 2-oxide.
Anuradha G, Gopalsamy V, Veera Reddy A, Laxminarasimhulu G. Anuradha G, et al. Acta Crystallogr Sect E Struct Rep Online. 2012 Oct 1;68(Pt 10):o2957. doi: 10.1107/S160053681203838X. Epub 2012 Sep 19. Acta Crystallogr Sect E Struct Rep Online. 2012. PMID: 23125740 Free PMC article.
The benzyl ring is inclined to the isoxazole ring by 74.19 (8) and is in a +sc conformation with respect to the benzisoxazole unit. In the crystal, C-H O hydrogen bonds link the mol-ecules, forming zigzag chains propagating along the b axis. ...
The benzyl ring is inclined to the isoxazole ring by 74.19 (8) and is in a +sc conformation with respect to the benzisoxazole unit. …
326 results