29662238 27919657 28395337 24708493 23149805 23580166 34648283 25993269 35566172 29330437 35611405 29349448 28032978 23033157 23586645 27240467 25529737 27107013 36517522 28657320 27976818 27870835 28506582 - Search Results

Year	Number of Results
2012	2
2013	2
2014	2
2015	2
2016	5
2017	7
2018	3
2021	1
2022	3
2023	0

1

Structural underpinnings of oestrogen receptor mutations in endocrine therapy resistance.

Katzenellenbogen JA, Mayne CG, Katzenellenbogen BS, Greene GL, Chandarlapaty S. Katzenellenbogen JA, et al. Nat Rev Cancer. 2018 Jun;18(6):377-388. doi: 10.1038/s41568-018-0001-z. Nat Rev Cancer. 2018. PMID: 29662238 Free PMC article. Review.

2

Synthesis of novel steroidal agonists, partial agonists, and antagonists for the glucocorticoid receptor.

Jin Z, Lin H, Srinivasan S, Nwachukwu JC, Bruno N, Griffin PR, Nettles KW, Kamenecka TM. Jin Z, et al. Bioorg Med Chem Lett. 2017 Jan 15;27(2):347-353. doi: 10.1016/j.bmcl.2016.11.007. Epub 2016 Nov 15. Bioorg Med Chem Lett. 2017. PMID: 27919657

3

Effects of vaginal conjugated equine estrogens and ospemifene on the rat vaginal wall and lower urinary tract.

Maldonado PA, Montoya TI, Acevedo JF, Keller PW, Word RA. Maldonado PA, et al. Biol Reprod. 2017 Jan 1;96(1):81-92. doi: 10.1095/biolreprod.116.144428. Biol Reprod. 2017. PMID: 28395337 Free PMC article.

4

Triaryl-substituted Schiff bases are high-affinity subtype-selective ligands for the estrogen receptor.

Liao ZQ, Dong C, Carlson KE, Srinivasan S, Nwachukwu JC, Chesnut RW, Sharma A, Nettles KW, Katzenellenbogen JA, Zhou HB. Liao ZQ, et al. J Med Chem. 2014 Apr 24;57(8):3532-45. doi: 10.1021/jm500268j. Epub 2014 Apr 7. J Med Chem. 2014. PMID: 24708493 Free PMC article.

5

Discovery of novel SERMs with a ferrocenyl entity based on the oxabicyclo[2.2.1]heptene scaffold and evaluation of their antiproliferative effects in breast cancer cells.

Zheng Y, Wang C, Li C, Qiao J, Zhang F, Huang M, Ren W, Dong C, Huang J, Zhou HB. Zheng Y, et al. Org Biomol Chem. 2012 Dec 28;10(48):9689-99. doi: 10.1039/c2ob26226f. Epub 2012 Nov 14. Org Biomol Chem. 2012. PMID: 23149805

6

Designer antiandrogens join the race against drug resistance.

Josan JS, Katzenellenbogen JA. Josan JS, et al. Elife. 2013 Apr 9;2:e00692. doi: 10.7554/eLife.00692. Elife. 2013. PMID: 23580166 Free PMC article.

7

Human Estrogen Receptor α Antagonists. Part 1: 3-D QSAR-Driven Rational Design of Innovative Coumarin-Related Antiestrogens as Breast Cancer Suppressants through Structure-Based and Ligand-Based Studies.

Mihović N, Tomašević N, Matić S, Mitrović MM, Kostić DA, Sabatino M, Antonini L, Ragno R, Mladenović M. Mihović N, et al. J Chem Inf Model. 2021 Oct 25;61(10):5028-5053. doi: 10.1021/acs.jcim.1c00530. Epub 2021 Oct 14. J Chem Inf Model. 2021. PMID: 34648283

8

Novel Bioactive Hybrid Compound Dual Targeting Estrogen Receptor and Histone Deacetylase for the Treatment of Breast Cancer.

Tang C, Li C, Zhang S, Hu Z, Wu J, Dong C, Huang J, Zhou HB. Tang C, et al. J Med Chem. 2015 Jun 11;58(11):4550-72. doi: 10.1021/acs.jmedchem.5b00099. Epub 2015 Jun 2. J Med Chem. 2015. PMID: 25993269

9

Human Estrogen Receptor Alpha Antagonists, Part 3: 3-D Pharmacophore and 3-D QSAR Guided Brefeldin A Hit-to-Lead Optimization toward New Breast Cancer Suppressants.

Kurtanović N, Tomašević N, Matić S, Proia E, Sabatino M, Antonini L, Mladenović M, Ragno R. Kurtanović N, et al. Molecules. 2022 Apr 28;27(9):2823. doi: 10.3390/molecules27092823. Molecules. 2022. PMID: 35566172 Free PMC article.

10

A Computational Assay of Estrogen Receptor α Antagonists Reveals the Key Common Structural Traits of Drugs Effectively Fighting Refractory Breast Cancers.

Pavlin M, Spinello A, Pennati M, Zaffaroni N, Gobbi S, Bisi A, Colombo G, Magistrato A. Pavlin M, et al. Sci Rep. 2018 Jan 12;8(1):649. doi: 10.1038/s41598-017-17364-4. Sci Rep. 2018. PMID: 29330437 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

Search Page

Search Results