29981240 27835801 31835873 27768894 28516479 28220706 30196704 36153039 33761251 31515283 28655732 33636308 28750804 28750807 26529344 27046127 27712124 - Search Results

Year	Number of Results
2015	1
2016	5
2017	6
2018	2
2019	3
2021	2
2022	1
2023	0

1

Allosteric and orthosteric pharmacology of cannabidiol and cannabidiol-dimethylheptyl at the type 1 and type 2 cannabinoid receptors.

Tham M, Yilmaz O, Alaverdashvili M, Kelly MEM, Denovan-Wright EM, Laprairie RB. Tham M, et al. Br J Pharmacol. 2019 May;176(10):1455-1469. doi: 10.1111/bph.14440. Epub 2018 Aug 10. Br J Pharmacol. 2019. PMID: 29981240 Free PMC article.

2

Cannabinoid receptor ligand bias: implications in the central nervous system.

Laprairie RB, Bagher AM, Denovan-Wright EM. Laprairie RB, et al. Curr Opin Pharmacol. 2017 Feb;32:32-43. doi: 10.1016/j.coph.2016.10.005. Epub 2016 Nov 9. Curr Opin Pharmacol. 2017. PMID: 27835801 Review.

3

Covalent Inhibition of the Histamine H₃ Receptor.

Wágner G, Mocking TAM, Kooistra AJ, Slynko I, Ábrányi-Balogh P, Keserű GM, Wijtmans M, Vischer HF, de Esch IJP, Leurs R. Wágner G, et al. Molecules. 2019 Dec 11;24(24):4541. doi: 10.3390/molecules24244541. Molecules. 2019. PMID: 31835873 Free PMC article.

4

Crystal Structure of the Human Cannabinoid Receptor CB₁.

Hua T, Vemuri K, Pu M, Qu L, Han GW, Wu Y, Zhao S, Shui W, Li S, Korde A, Laprairie RB, Stahl EL, Ho JH, Zvonok N, Zhou H, Kufareva I, Wu B, Zhao Q, Hanson MA, Bohn LM, Makriyannis A, Stevens RC, Liu ZJ. Hua T, et al. Cell. 2016 Oct 20;167(3):750-762.e14. doi: 10.1016/j.cell.2016.10.004. Cell. 2016. PMID: 27768894 Free PMC article.

5

Gα_s signalling of the CB₁ receptor and the influence of receptor number.

Finlay DB, Cawston EE, Grimsey NL, Hunter MR, Korde A, Vemuri VK, Makriyannis A, Glass M. Finlay DB, et al. Br J Pharmacol. 2017 Aug;174(15):2545-2562. doi: 10.1111/bph.13866. Epub 2017 Jun 19. Br J Pharmacol. 2017. PMID: 28516479 Free PMC article.

6

Human Cannabinoid Receptor 2 Ligand-Interaction Motif: Transmembrane Helix 2 Cysteine, C2.59(89), as Determinant of Classical Cannabinoid Agonist Activity and Binding Pose.

Zhou H, Peng Y, Halikhedkar A, Fan P, Janero DR, Thakur GA, Mercier RW, Sun X, Ma X, Makriyannis A. Zhou H, et al. ACS Chem Neurosci. 2017 Jun 21;8(6):1338-1347. doi: 10.1021/acschemneuro.7b00003. Epub 2017 Mar 1. ACS Chem Neurosci. 2017. PMID: 28220706

7

( R)- N-(1-Methyl-2-hydroxyethyl)-13-( S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes.

Liu Y, Ji L, Eno M, Kudalkar S, Li AL, Schimpgen M, Benchama O, Morales P, Xu S, Hurst D, Wu S, Mohammad KA, Wood JT, Zvonok N, Papahatjis DP, Zhou H, Honrao C, Mackie K, Reggio P, Hohmann AG, Marnett LJ, Makriyannis A, Nikas SP. Liu Y, et al. J Med Chem. 2018 Oct 11;61(19):8639-8657. doi: 10.1021/acs.jmedchem.8b00611. Epub 2018 Sep 21. J Med Chem. 2018. PMID: 30196704

8

Differential Enantiomer-Specific Signaling of Cannabidiol at CB₁ Receptors.

Bosquez-Berger T, Wilson S, Iliopoulos-Tsoutsouvas C, Jiang S, Wager-Miller J, Nikas SP, Mackie KP, Makriyannis A, Straiker A. Bosquez-Berger T, et al. Mol Pharmacol. 2022 Dec;102(6):259-268. doi: 10.1124/molpharm.121.000305. Epub 2022 Sep 24. Mol Pharmacol. 2022. PMID: 36153039

9

Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists.

Jiang S, Iliopoulos-Tsoutsouvas C, Tong F, Brust CA, Keenan CM, Raghav JG, Hua T, Wu S, Ho JH, Wu Y, Grim TW, Zvonok N, Thakur GA, Liu ZJ, Sharkey KA, Bohn LM, Nikas SP, Makriyannis A. Jiang S, et al. J Med Chem. 2021 Apr 8;64(7):3870-3884. doi: 10.1021/acs.jmedchem.0c02053. Epub 2021 Mar 24. J Med Chem. 2021. PMID: 33761251

10

Probing the CB₁ Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist.

Laprairie RB, Vemuri K, Stahl EL, Korde A, Ho JH, Grim TW, Hua T, Wu Y, Stevens RC, Liu ZJ, Makriyannis A, Bohn LM. Laprairie RB, et al. Mol Pharmacol. 2019 Nov;96(5):619-628. doi: 10.1124/mol.119.116483. Epub 2019 Sep 12. Mol Pharmacol. 2019. PMID: 31515283 Free PMC article.

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