31038398 30833575 29662238 28514424 33965842 35566172 35955864 29330437 30831350 34452998 28514419 29783894 29915250 28032978 29152682 28954197 30731397 30123887 31289329 28770632 33479648 30939353 28657320 31175940 30053783 30108860 28754571 3548730 - Search Results

Year	Number of Results
2016	1
2017	11
2018	8
2019	11
2020	5
2021	2
2022	4
2023	0

1

Evaluation of binding and antagonism/downregulation of brilanestrant molecule in estrogen receptor-α via quantum mechanics/molecular mechanics, molecular dynamics and binding free energy calculations.

Chinnasamy K, Saravanan M, Poomani K. Chinnasamy K, et al. J Biomol Struct Dyn. 2020 Jan;38(1):219-235. doi: 10.1080/07391102.2019.1574605. Epub 2019 Apr 30. J Biomol Struct Dyn. 2020. PMID: 31038398

2

Pocket similarity identifies selective estrogen receptor modulators as microtubule modulators at the taxane site.

Lo YC, Cormier O, Liu T, Nettles KW, Katzenellenbogen JA, Stearns T, Altman RB. Lo YC, et al. Nat Commun. 2019 Mar 4;10(1):1033. doi: 10.1038/s41467-019-08965-w. Nat Commun. 2019. PMID: 30833575 Free PMC article.

3

Structural underpinnings of oestrogen receptor mutations in endocrine therapy resistance.

Katzenellenbogen JA, Mayne CG, Katzenellenbogen BS, Greene GL, Chandarlapaty S. Katzenellenbogen JA, et al. Nat Rev Cancer. 2018 Jun;18(6):377-388. doi: 10.1038/s41568-018-0001-z. Nat Rev Cancer. 2018. PMID: 29662238 Free PMC article. Review.

4

Corrigendum: Full antagonism of the estrogen receptor without a prototypical ligand side chain.

Srinivasan S, Nwachukwu JC, Bruno NE, Dharmarajan V, Goswami D, Kastrati I, Novick S, Nowak J, Cavett V, Zhou HB, Boonmuen N, Zhao Y, Min J, Frasor J, Katzenellenbogen BS, Griffin PR, Katzenellenbogen JA, Nettles KW. Srinivasan S, et al. Nat Chem Biol. 2017 May 17;13(6):691. doi: 10.1038/nchembio0617-691c. Nat Chem Biol. 2017. PMID: 28514424 No abstract available.

5

Novel hybrid conjugates with dual estrogen receptor α degradation and histone deacetylase inhibitory activities for breast cancer therapy.

Zhao C, Tang C, Li C, Ning W, Hu Z, Xin L, Zhou HB, Huang J. Zhao C, et al. Bioorg Med Chem. 2021 Jun 15;40:116185. doi: 10.1016/j.bmc.2021.116185. Epub 2021 May 1. Bioorg Med Chem. 2021. PMID: 33965842

6

Human Estrogen Receptor Alpha Antagonists, Part 3: 3-D Pharmacophore and 3-D QSAR Guided Brefeldin A Hit-to-Lead Optimization toward New Breast Cancer Suppressants.

Kurtanović N, Tomašević N, Matić S, Proia E, Sabatino M, Antonini L, Mladenović M, Ragno R. Kurtanović N, et al. Molecules. 2022 Apr 28;27(9):2823. doi: 10.3390/molecules27092823. Molecules. 2022. PMID: 35566172 Free PMC article.

7

Exploring Ligand Binding Domain Dynamics in the NRs Superfamily.

D'Arrigo G, Autiero I, Gianquinto E, Siragusa L, Baroni M, Cruciani G, Spyrakis F. D'Arrigo G, et al. Int J Mol Sci. 2022 Aug 5;23(15):8732. doi: 10.3390/ijms23158732. Int J Mol Sci. 2022. PMID: 35955864 Free PMC article.

8

A Computational Assay of Estrogen Receptor α Antagonists Reveals the Key Common Structural Traits of Drugs Effectively Fighting Refractory Breast Cancers.

Pavlin M, Spinello A, Pennati M, Zaffaroni N, Gobbi S, Bisi A, Colombo G, Magistrato A. Pavlin M, et al. Sci Rep. 2018 Jan 12;8(1):649. doi: 10.1038/s41598-017-17364-4. Sci Rep. 2018. PMID: 29330437 Free PMC article.

9

Computational insights on agonist and antagonist mechanisms of estrogen receptor α induced by bisphenol A analogues.

Cao H, Wang L, Cao M, Ye T, Sun Y. Cao H, et al. Environ Pollut. 2019 May;248:536-545. doi: 10.1016/j.envpol.2019.02.058. Epub 2019 Feb 22. Environ Pollut. 2019. PMID: 30831350

10

Dual-mechanism estrogen receptor inhibitors.

Min J, Nwachukwu JC, Min CK, Njeri JW, Srinivasan S, Rangarajan ES, Nettles CC, Sanabria Guillen V, Ziegler Y, Yan S, Carlson KE, Hou Y, Kim SH, Novick S, Pascal BD, Houtman R, Griffin PR, Izard T, Katzenellenbogen BS, Katzenellenbogen JA, Nettles KW. Min J, et al. Proc Natl Acad Sci U S A. 2021 Aug 31;118(35):e2101657118. doi: 10.1073/pnas.2101657118. Proc Natl Acad Sci U S A. 2021. PMID: 34452998 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

Search Page

Search Results