Three-dimensional quantitative structure-activity relationship analyses using comparative molecular field analysis and comparative molecular similarity indices analysis to elucidate selectivity differences of inhibitors binding to trypsin, thrombin, and factor Xa.
J Med Chem. 1999 Feb 11;42(3):458-77. doi: 10.1021/jm981062r.
J Med Chem. 1999.
PMID: 9986717