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Structure-Bioactivity Relationships of Lapatinib Derived Analogs against Schistosoma mansoni.
ACS Med Chem Lett. 2020 Jan 10;11(3):258-265. doi: 10.1021/acsmedchemlett.9b00455. eCollection 2020 Mar 12.
ACS Med Chem Lett. 2020.
PMID: 32184954
Free PMC article.
Scaffold and Parasite Hopping: Discovery of New Protozoal Proliferation Inhibitors.
Singh B, Bernatchez JA, McCall LI, Calvet CM, Ackermann J, Souza JM, Thomas D, Silva EM, Bachovchin KA, Klug DM, Jalani HB, Bag S, Buskes MJ, Leed SE, Roncal NE, Penn EC, Erath J, Rodriguez A, Sciotti RJ, Campbell RF, McKerrow J, Siqueira-Neto JL, Ferrins L, Pollastri MP.
Singh B, et al. Among authors: bachovchin ka.
ACS Med Chem Lett. 2020 Jan 10;11(3):249-257. doi: 10.1021/acsmedchemlett.9b00453. eCollection 2020 Mar 12.
ACS Med Chem Lett. 2020.
PMID: 32184953
Free PMC article.
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Improvement of Aqueous Solubility of Lapatinib-Derived Analogues: Identification of a Quinolinimine Lead for Human African Trypanosomiasis Drug Development.
Bachovchin KA, Sharma A, Bag S, Klug DM, Schneider KM, Singh B, Jalani HB, Buskes MJ, Mehta N, Tanghe S, Momper JD, Sciotti RJ, Rodriguez A, Mensa-Wilmot K, Pollastri MP, Ferrins L.
Bachovchin KA, et al.
J Med Chem. 2019 Jan 24;62(2):665-687. doi: 10.1021/acs.jmedchem.8b01365. Epub 2019 Jan 10.
J Med Chem. 2019.
PMID: 30565932
Free PMC article.
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Corrigendum to "Optimization of physicochemical properties for 4-Anilinoquinazoline inhibitors of trypanosome proliferation" [Eur. J. Med. Chem. 141 (2017) 446-459].
Woodring JL, Bachovchin KA, Brady KG, Gallerstein MF, Erath J, Tanghe S, Leed SE, Rodriguez A, Mensa-Wilmot K, Sciotti RJ, Pollastri MP.
Woodring JL, et al. Among authors: bachovchin ka.
Eur J Med Chem. 2018 May 25;152:515. doi: 10.1016/j.ejmech.2018.05.002. Epub 2018 May 10.
Eur J Med Chem. 2018.
PMID: 29754075
No abstract available.
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Optimization of physicochemical properties for 4-anilinoquinazoline inhibitors of trypanosome proliferation.
Woodring JL, Bachovchin KA, Brady KG, Gallerstein MF, Erath J, Tanghe S, Leed SE, Rodriguez A, Mensa-Wilmot K, Sciotti RJ, Pollastri MP.
Woodring JL, et al. Among authors: bachovchin ka.
Eur J Med Chem. 2017 Dec 1;141:446-459. doi: 10.1016/j.ejmech.2017.10.007. Epub 2017 Oct 6.
Eur J Med Chem. 2017.
PMID: 29049963
Free PMC article.
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Antiparasitic Lead Discovery: Toward Optimization of a Chemotype with Activity Against Multiple Protozoan Parasites.
Devine W, Thomas SM, Erath J, Bachovchin KA, Lee PJ, Leed SE, Rodriguez A, Sciotti RJ, Mensa-Wilmot K, Pollastri MP.
Devine W, et al. Among authors: bachovchin ka.
ACS Med Chem Lett. 2017 Feb 5;8(3):350-354. doi: 10.1021/acsmedchemlett.7b00011. eCollection 2017 Mar 9.
ACS Med Chem Lett. 2017.
PMID: 28337329
Free PMC article.
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Identifying bias in CCR1 antagonists using radiolabelled binding, receptor internalization, β-arrestin translocation and chemotaxis assays.
Gilchrist A, Gauntner TD, Fazzini A, Alley KM, Pyen DS, Ahn J, Ha SJ, Willett A, Sansom SE, Yarfi JL, Bachovchin KA, Mazzoni MR, Merritt JR.
Gilchrist A, et al. Among authors: bachovchin ka.
Br J Pharmacol. 2014 Nov;171(22):5127-38. doi: 10.1111/bph.12835.
Br J Pharmacol. 2014.
PMID: 24990525
Free PMC article.
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