Barczyk A - Search Results

1

Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure.

Boulahjar R, Rincon Arias A, Bolteau R, Renault N, Coevoet M, Barczyk A, Duroux R, Yous S, Melnyk P, Agouridas L. Boulahjar R, et al. Among authors: barczyk a. Bioorg Med Chem. 2018 Jul 23;26(12):3296-3307. doi: 10.1016/j.bmc.2018.04.057. Epub 2018 Apr 30. Bioorg Med Chem. 2018. PMID: 29753566 Free article.

2

Switching cannabinoid response from CB(2) agonists to FAAH inhibitors.

Tourteau A, Leleu-Chavain N, Body-Malapel M, Andrzejak V, Barczyk A, Djouina M, Rigo B, Desreumaux P, Chavatte P, Millet R. Tourteau A, et al. Among authors: barczyk a. Bioorg Med Chem Lett. 2014 Mar 1;24(5):1322-6. doi: 10.1016/j.bmcl.2014.01.056. Epub 2014 Jan 28. Bioorg Med Chem Lett. 2014. PMID: 24508127

3

Inhibition of tumor cell growth and angiogenesis by 7-aminoalkoxy-4-aryloxy-quinazoline ureas, a novel series of multi-tyrosine kinase inhibitors.

Ravez S, Barczyk A, Six P, Cagnon A, Garofalo A, Goossens L, Depreux P. Ravez S, et al. Among authors: barczyk a. Eur J Med Chem. 2014 May 22;79:369-81. doi: 10.1016/j.ejmech.2014.04.007. Epub 2014 Apr 5. Eur J Med Chem. 2014. PMID: 24747748

4

Conformational Restriction Leading to a Selective CB2 Cannabinoid Receptor Agonist Orally Active Against Colitis.

El Bakali J, Muccioli GG, Body-Malapel M, Djouina M, Klupsch F, Ghinet A, Barczyk A, Renault N, Chavatte P, Desreumaux P, Lambert DM, Millet R. El Bakali J, et al. Among authors: barczyk a. ACS Med Chem Lett. 2014 Dec 4;6(2):198-203. doi: 10.1021/ml500439x. eCollection 2015 Feb 12. ACS Med Chem Lett. 2014. PMID: 25699149 Free PMC article.

5

Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors.

Ravez S, Arsenlis S, Barczyk A, Dupont A, Frédérick R, Hesse S, Kirsch G, Depreux P, Goossens L. Ravez S, et al. Among authors: barczyk a. Bioorg Med Chem. 2015 Nov 15;23(22):7340-7. doi: 10.1016/j.bmc.2015.10.035. Epub 2015 Oct 24. Bioorg Med Chem. 2015. PMID: 26526740

6

Synthesis of triazoloquinazolinone based compounds as tubulin polymerization inhibitors and vascular disrupting agents.

Driowya M, Leclercq J, Verones V, Barczyk A, Lecoeur M, Renault N, Flouquet N, Ghinet A, Berthelot P, Lebegue N. Driowya M, et al. Among authors: barczyk a. Eur J Med Chem. 2016 Jun 10;115:393-405. doi: 10.1016/j.ejmech.2016.03.056. Epub 2016 Mar 22. Eur J Med Chem. 2016. PMID: 27031215

7

Design, synthesis and biological evaluation of potent FAAH inhibitors.

Tuo W, Leleu-Chavain N, Barczyk A, Renault N, Lemaire L, Chavatte P, Millet R. Tuo W, et al. Among authors: barczyk a. Bioorg Med Chem Lett. 2016 Jun 1;26(11):2701-5. doi: 10.1016/j.bmcl.2016.04.004. Epub 2016 Apr 23. Bioorg Med Chem Lett. 2016. PMID: 27117424

8

Synthesis and Biological Evaluation of N-[2-(4-Hydroxyphenylamino)-pyridin-3-yl]-4-methoxy-benzenesulfonamide (ABT-751) Tricyclic Analogues as Antimitotic and Antivascular Agents with Potent in Vivo Antitumor Activity.

Segaoula Z, Leclercq J, Verones V, Flouquet N, Lecoeur M, Ach L, Renault N, Barczyk A, Melnyk P, Berthelot P, Thuru X, Lebegue N. Segaoula Z, et al. Among authors: barczyk a. J Med Chem. 2016 Sep 22;59(18):8422-40. doi: 10.1021/acs.jmedchem.6b00847. Epub 2016 Aug 30. J Med Chem. 2016. PMID: 27538123 Free article.

9

Synthesis and pharmacological evaluation of benzamide derivatives as potent and selective sigma-1 protein ligands.

Donnier-Maréchal M, Carato P, Larchanché PE, Ravez S, Boulahjar R, Barczyk A, Oxombre B, Vermersch P, Melnyk P. Donnier-Maréchal M, et al. Among authors: barczyk a. Eur J Med Chem. 2017 Sep 29;138:964-978. doi: 10.1016/j.ejmech.2017.07.014. Epub 2017 Jul 12. Eur J Med Chem. 2017. PMID: 28756263

10

Development of novel oxazolo[5,4-d]pyrimidines as competitive CB₂ neutral antagonists based on scaffold hopping.

Tuo W, Bollier M, Leleu-Chavain N, Lemaire L, Barczyk A, Dezitter X, Klupsch F, Szczepanski F, Spencer J, Chavatte P, Millet R. Tuo W, et al. Among authors: barczyk a. Eur J Med Chem. 2018 Feb 25;146:68-78. doi: 10.1016/j.ejmech.2018.01.034. Epub 2018 Jan 16. Eur J Med Chem. 2018. PMID: 29360044

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