Chemoproteomic discovery of a brain-penetrant, covalent NLRP3 inhibitor that binds a novel allosteric pocket.
Rogness DC, Sievert EP, Vartabedian VF, Bernard SM, Aitchison E, Tao W, Lindvall M, Qian J, Eissler CL, Nordin BE, Horning BD, Kingston C, Lamb KN, Bell JC, Lu B, Pollock J, Shi J, Khattri R, Weinstein DS, Patricelli MP, Cook BN, Simon GM.
Rogness DC, et al. Among authors: bell jc.
Br J Pharmacol. 2026 Aug 8. doi: 10.1111/bph.70626. Online ahead of print.
Br J Pharmacol. 2026.
PMID: 42569816