SuFEx-based antitubercular compound irreversibly inhibits Pks13.
Krieger IV, Sukheja P, Yang B, Tang S, Selle D, Woods A, Engelhart C, Kumar P, Harbut MB, Liu D, Tsuda B, Qin B, Bare GAL, Li G, Chi V, Gambacurta J, Hvizdos J, Reagan M, Jones IL, Massoudi LM, Woolhiser LK, Cascioferro A, Kundrick E, Singh P, Reiley W, Ioerger TR, Kandula DR, McCabe JW, Guo T, Alland D, Boshoff HI, Schnappinger D, Robertson GT, Mdluli K, Lee KJ, Dong J, Li S, Schultz PG, Joseph SB, Love MS, Sharpless KB, Petrassi HM, Chatterjee AK, Sacchettini JC, McNamara CW.
Krieger IV, et al. Among authors: qin b.
Nature. 2025 Sep;645(8081):755-763. doi: 10.1038/s41586-025-09286-3. Epub 2025 Jul 30.
Nature. 2025.
PMID: 40739353