Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
8 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Crystal structures of anaplastic lymphoma kinase in complex with ATP competitive inhibitors.
Biochemistry. 2010 Aug 17;49(32):6813-25. doi: 10.1021/bi1005514.
Biochemistry. 2010.
PMID: 20695522
Discovery of Entrectinib: A New 3-Aminoindazole As a Potent Anaplastic Lymphoma Kinase (ALK), c-ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor.
Menichincheri M, Ardini E, Magnaghi P, Avanzi N, Banfi P, Bossi R, Buffa L, Canevari G, Ceriani L, Colombo M, Corti L, Donati D, Fasolini M, Felder E, Fiorelli C, Fiorentini F, Galvani A, Isacchi A, Borgia AL, Marchionni C, Nesi M, Orrenius C, Panzeri A, Pesenti E, Rusconi L, Saccardo MB, Vanotti E, Perrone E, Orsini P.
Menichincheri M, et al. Among authors: borgia al.
J Med Chem. 2016 Apr 14;59(7):3392-408. doi: 10.1021/acs.jmedchem.6b00064. Epub 2016 Mar 30.
J Med Chem. 2016.
PMID: 27003761
Item in Clipboard
The TPM3-NTRK1 rearrangement is a recurring event in colorectal carcinoma and is associated with tumor sensitivity to TRKA kinase inhibition.
Ardini E, Bosotti R, Borgia AL, De Ponti C, Somaschini A, Cammarota R, Amboldi N, Raddrizzani L, Milani A, Magnaghi P, Ballinari D, Casero D, Gasparri F, Banfi P, Avanzi N, Saccardo MB, Alzani R, Bandiera T, Felder E, Donati D, Pesenti E, Sartore-Bianchi A, Gambacorta M, Pierotti MA, Siena S, Veronese S, Galvani A, Isacchi A.
Ardini E, et al. Among authors: borgia al.
Mol Oncol. 2014 Dec;8(8):1495-507. doi: 10.1016/j.molonc.2014.06.001. Epub 2014 Jun 12.
Mol Oncol. 2014.
PMID: 24962792
Free PMC article.
Item in Clipboard
Correction to Discovery of Entrectinib: A New 3-Aminoindazole as a Potent Anaplastic Lymphoma Kinase (ALK), c-ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor.
Menichincheri M, Ardini E, Magnaghi P, Avanzi N, Banfi P, Bossi R, Buffa L, Canevari G, Ceriani L, Colombo M, Corti L, Donati D, Fasolini M, Felder E, Fiorelli C, Fiorentini F, Galvani A, Isacchi A, Borgia AL, Marchionni C, Nesi M, Orrenius C, Panzeri A, Pesenti E, Rusconi L, Saccardo MB, Vanotti E, Perrone E, Orsini P.
Menichincheri M, et al. Among authors: borgia al.
J Med Chem. 2019 Sep 12;62(17):8364. doi: 10.1021/acs.jmedchem.9b01259. Epub 2019 Aug 19.
J Med Chem. 2019.
PMID: 31424209
No abstract available.
Item in Clipboard
Synthesis and binding mode of heterocyclic analogues of suramin inhibiting the human basic fibroblast growth factor.
Manetti F, Cappello V, Botta M, Corelli F, Mongelli N, Biasoli G, Borgia AL, Ciomei M.
Manetti F, et al. Among authors: borgia al.
Bioorg Med Chem. 1998 Jul;6(7):947-58. doi: 10.1016/s0968-0896(98)00052-2.
Bioorg Med Chem. 1998.
PMID: 9730230
Item in Clipboard
Research on anti-HIV-1 agents. Investigation on the CD4-Suradista binding mode through docking experiments.
Manetti F, Corelli F, Mongelli N, Borgia AL, Botta M.
Manetti F, et al. Among authors: borgia al.
J Comput Aided Mol Des. 2000 May;14(4):355-68. doi: 10.1023/a:1008154931914.
J Comput Aided Mol Des. 2000.
PMID: 10815772
Item in Clipboard
Novel sulfonated and phosphonated analogs of distamycin which inhibit the replication of HIV.
Clanton DJ, Buckheit RW Jr, Terpening SJ, Kiser R, Mongelli N, Borgia AL, Schultz R, Narayanan V, Bader JP, Rice WG.
Clanton DJ, et al. Among authors: borgia al.
Antiviral Res. 1995 Aug;27(4):335-54. doi: 10.1016/0166-3542(95)00017-g.
Antiviral Res. 1995.
PMID: 8540754
Item in Clipboard
Trial of Anifrolumab in Active Systemic Lupus Erythematosus.
Morand EF, Furie R, Tanaka Y, Bruce IN, Askanase AD, Richez C, Bae SC, Brohawn PZ, Pineda L, Berglind A, Tummala R; TULIP-2 Trial Investigators.
Morand EF, et al.
N Engl J Med. 2020 Jan 16;382(3):211-221. doi: 10.1056/NEJMoa1912196. Epub 2019 Dec 18.
N Engl J Med. 2020.
PMID: 31851795
Clinical Trial.
Item in Clipboard
Cite
Cite