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Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors.
ChemMedChem. 2020 Jun 4;15(11):955-960. doi: 10.1002/cmdc.202000007. Epub 2020 Apr 6.
ChemMedChem. 2020.
PMID: 32181984
Make the right measurement: Discovery of an allosteric inhibition site for p300-HAT.
Gardberg AS, Huhn AJ, Cummings R, Bommi-Reddy A, Poy F, Setser J, Vivat V, Brucelle F, Wilson J.
Gardberg AS, et al. Among authors: brucelle f.
Struct Dyn. 2019 Oct 11;6(5):054702. doi: 10.1063/1.5119336. eCollection 2019 Sep.
Struct Dyn. 2019.
PMID: 31649965
Free PMC article.
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Discovery of CPI-1612: A Potent, Selective, and Orally Bioavailable EP300/CBP Histone Acetyltransferase Inhibitor.
Wilson JE, Patel G, Patel C, Brucelle F, Huhn A, Gardberg AS, Poy F, Cantone N, Bommi-Reddy A, Sims RJ 3rd, Cummings RT, Levell JR.
Wilson JE, et al. Among authors: brucelle f.
ACS Med Chem Lett. 2020 Apr 23;11(6):1324-1329. doi: 10.1021/acsmedchemlett.0c00155. eCollection 2020 Jun 11.
ACS Med Chem Lett. 2020.
PMID: 32551019
Free PMC article.
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Design and Synthesis of Styrenylcyclopropylamine LSD1 Inhibitors.
Gehling VS, McGrath JP, Duplessis M, Khanna A, Brucelle F, Vaswani RG, Côté A, Stuckey J, Watson V, Cummings RT, Balasubramanian S, Iyer P, Sawant P, Good AC, Albrecht BK, Harmange JC, Audia JE, Bellon SF, Trojer P, Levell JR.
Gehling VS, et al. Among authors: brucelle f.
ACS Med Chem Lett. 2020 May 6;11(6):1213-1220. doi: 10.1021/acsmedchemlett.0c00060. eCollection 2020 Jun 11.
ACS Med Chem Lett. 2020.
PMID: 32551003
Free PMC article.
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Preparation of the Core Structure of Aspidosperma and Strychnos Alkaloids from Aryl Azides by a Cascade Radical Cyclization.
Wyler B, Brucelle F, Renaud P.
Wyler B, et al. Among authors: brucelle f.
Org Lett. 2016 Mar 18;18(6):1370-3. doi: 10.1021/acs.orglett.6b00306. Epub 2016 Feb 29.
Org Lett. 2016.
PMID: 26926777
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Synthesis of a leucomitosane via a diastereoselective radical cascade.
Brucelle F, Renaud P.
Brucelle F, et al.
J Org Chem. 2013 Jun 21;78(12):6245-52. doi: 10.1021/jo4009904. Epub 2013 Jun 7.
J Org Chem. 2013.
PMID: 23721078
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Synthesis of indolines, indoles, and benzopyrrolizidinones from simple aryl azides.
Brucelle F, Renaud P.
Brucelle F, et al.
Org Lett. 2012 Jun 15;14(12):3048-51. doi: 10.1021/ol301120w. Epub 2012 May 30.
Org Lett. 2012.
PMID: 22646529
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