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Design and synthesis of novel indole beta-diketo acid derivatives as HIV-1 integrase inhibitors.
Sechi M, Derudas M, Dallocchio R, Dessì A, Bacchi A, Sannia L, Carta F, Palomba M, Ragab O, Chan C, Shoemaker R, Sei S, Dayam R, Neamati N. Sechi M, et al. J Med Chem. 2004 Oct 7;47(21):5298-310. doi: 10.1021/jm049944f. J Med Chem. 2004. PMID: 15456274
To establish a coherent structure-activity relationship among the substituted indole nucleus bearing a beta-diketo acid moiety, a series of substituted indole-beta-diketo acids (4a-f and 5a-e) were synthesized. ...
To establish a coherent structure-activity relationship among the substituted indole nucleus bearing a beta-diketo acid moiety, a series of …
From ligand to complexes. Part 2. Remarks on human immunodeficiency virus type 1 integrase inhibition by beta-diketo acid metal complexes.
Bacchi A, Biemmi M, Carcelli M, Carta F, Compari C, Fisicaro E, Rogolino D, Sechi M, Sippel M, Sotriffer CA, Sanchez TW, Neamati N. Bacchi A, et al. J Med Chem. 2008 Nov 27;51(22):7253-64. doi: 10.1021/jm800893q. J Med Chem. 2008. PMID: 18983138
Carbonic anhydrase inhibitors: inhibition of cytosolic carbonic anhydrase isozymes II and VII with simple aromatic sulfonamides and some azo dyes.
Carta F, Pothen B, Maresca A, Tiwari M, Singh V, Supuran CT. Carta F, et al. Chem Biol Drug Des. 2009 Aug;74(2):196-202. doi: 10.1111/j.1747-0285.2009.00842.x. Epub 2009 Jun 22. Chem Biol Drug Des. 2009. PMID: 19549076
Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides.
Maresca A, Carta F, Vullo D, Scozzafava A, Supuran CT. Maresca A, et al. Bioorg Med Chem Lett. 2009 Sep 1;19(17):4929-32. doi: 10.1016/j.bmcl.2009.07.088. Epub 2009 Jul 22. Bioorg Med Chem Lett. 2009. PMID: 19651511
Carbonic anhydrase inhibitors. Diazenylbenzenesulfonamides are potent and selective inhibitors of the tumor-associated isozymes IX and XII over the cytosolic isoforms I and II.
Carta F, Maresca A, Scozzafava A, Vullo D, Supuran CT. Carta F, et al. Bioorg Med Chem. 2009 Oct 15;17(20):7093-9. doi: 10.1016/j.bmc.2009.09.003. Epub 2009 Sep 6. Bioorg Med Chem. 2009. PMID: 19773173
Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.
Carta F, Maresca A, Covarrubias AS, Mowbray SL, Jones TA, Supuran CT. Carta F, et al. Bioorg Med Chem Lett. 2009 Dec 1;19(23):6649-54. doi: 10.1016/j.bmcl.2009.10.009. Epub 2009 Oct 7. Bioorg Med Chem Lett. 2009. PMID: 19846301
The β-carbonic anhydrases from Mycobacterium tuberculosis as drug targets.
Nishimori I, Minakuchi T, Maresca A, Carta F, Scozzafava A, Supuran CT. Nishimori I, et al. Curr Pharm Des. 2010;16(29):3300-9. doi: 10.2174/138161210793429814. Curr Pharm Des. 2010. PMID: 20819064 Review.
Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides.
Pacchiano F, Carta F, Vullo D, Scozzafava A, Supuran CT. Pacchiano F, et al. Bioorg Med Chem Lett. 2011 Jan 1;21(1):102-5. doi: 10.1016/j.bmcl.2010.11.064. Epub 2010 Nov 20. Bioorg Med Chem Lett. 2011. PMID: 21145236
Ureido-substituted benzenesulfonamides potently inhibit carbonic anhydrase IX and show antimetastatic activity in a model of breast cancer metastasis.
Pacchiano F, Carta F, McDonald PC, Lou Y, Vullo D, Scozzafava A, Dedhar S, Supuran CT. Pacchiano F, et al. J Med Chem. 2011 Mar 24;54(6):1896-902. doi: 10.1021/jm101541x. Epub 2011 Mar 1. J Med Chem. 2011. PMID: 21361354
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