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Conformationally restrained analogues of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor.
J Med Chem. 1992 Jan;35(1):124-35. doi: 10.1021/jm00079a016.
J Med Chem. 1992.
PMID: 1732519
Pravadoline: profile in isolated tissue preparations.
Ward SJ, Mastriani D, Casiano F, Arnold R.
Ward SJ, et al.
J Pharmacol Exp Ther. 1990 Dec;255(3):1230-9.
J Pharmacol Exp Ther. 1990.
PMID: 2175798
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Putative aminoalkylindoles (AAI) antagonists.
Casiano FM, Arnold R, Haycock D, Kuster J, Ward SJ.
Casiano FM, et al.
NIDA Res Monogr. 1990;105:295-6.
NIDA Res Monogr. 1990.
PMID: 1876017
No abstract available.
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WIN 64821, a novel neurokinin antagonist produced by an Aspergillus sp. II. Biological activity.
Oleynek JJ, Sedlock DM, Barrow CJ, Appell KC, Casiano F, Haycock D, Ward SJ, Kaplita P, Gillum AM.
Oleynek JJ, et al.
J Antibiot (Tokyo). 1994 Apr;47(4):399-410. doi: 10.7164/antibiotics.47.399.
J Antibiot (Tokyo). 1994.
PMID: 7515038
Free article.
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The nonpeptide WIN 64338 is a bradykinin B2 receptor antagonist.
Sawutz DG, Salvino JM, Dolle RE, Casiano F, Ward SJ, Houck WT, Faunce DM, Douty BD, Baizman E, Awad MM, et al.
Sawutz DG, et al.
Proc Natl Acad Sci U S A. 1994 May 24;91(11):4693-7. doi: 10.1073/pnas.91.11.4693.
Proc Natl Acad Sci U S A. 1994.
PMID: 8197121
Free PMC article.
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Aminoalkylindoles: actions on specific G-protein-linked receptors.
Pacheco M, Childers SR, Arnold R, Casiano F, Ward SJ.
Pacheco M, et al.
J Pharmacol Exp Ther. 1991 Apr;257(1):170-83.
J Pharmacol Exp Ther. 1991.
PMID: 1902257
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