De Logu A - Search Results

1

Improved BM212 MmpL3 inhibitor analogue shows efficacy in acute murine model of tuberculosis infection.

Poce G, Bates RH, Alfonso S, Cocozza M, Porretta GC, Ballell L, Rullas J, Ortega F, De Logu A, Agus E, La Rosa V, Pasca MR, De Rossi E, Wae B, Franzblau SG, Manetti F, Botta M, Biava M. Poce G, et al. Among authors: de logu a, de rossi e. PLoS One. 2013;8(2):e56980. doi: 10.1371/journal.pone.0056980. Epub 2013 Feb 21. PLoS One. 2013. PMID: 23437287 Free PMC article.

2

Ligand-based virtual screening, parallel solution-phase and microwave-assisted synthesis as tools to identify and synthesize new inhibitors of mycobacterium tuberculosis.

Manetti F, Magnani M, Castagnolo D, Passalacqua L, Botta M, Corelli F, Saddi M, Deidda D, De Logu A. Manetti F, et al. Among authors: de logu a. ChemMedChem. 2006 Sep;1(9):973-89. doi: 10.1002/cmdc.200600026. ChemMedChem. 2006. PMID: 16892466

3

1,5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings.

Biava M, Porretta GC, Poce G, De Logu A, Saddi M, Meleddu R, Manetti F, De Rossi E, Botta M. Biava M, et al. Among authors: de logu a, de rossi e. J Med Chem. 2008 Jun 26;51(12):3644-8. doi: 10.1021/jm701560p. J Med Chem. 2008. PMID: 18494459

4

Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis.

Castagnolo D, De Logu A, Radi M, Bechi B, Manetti F, Magnani M, Supino S, Meleddu R, Chisu L, Botta M. Castagnolo D, et al. Among authors: de logu a. Bioorg Med Chem. 2008 Sep 15;16(18):8587-91. doi: 10.1016/j.bmc.2008.08.016. Epub 2008 Aug 7. Bioorg Med Chem. 2008. PMID: 18752962 Free article.

5

Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis.

Castagnolo D, Radi M, Dessì F, Manetti F, Saddi M, Meleddu R, De Logu A, Botta M. Castagnolo D, et al. Among authors: de logu a. Bioorg Med Chem Lett. 2009 Apr 15;19(8):2203-5. doi: 10.1016/j.bmcl.2009.02.101. Epub 2009 Feb 28. Bioorg Med Chem Lett. 2009. PMID: 19299129

6

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones.

Castagnolo D, Manetti F, Radi M, Bechi B, Pagano M, De Logu A, Meleddu R, Saddi M, Botta M. Castagnolo D, et al. Among authors: de logu a. Bioorg Med Chem. 2009 Aug 1;17(15):5716-21. doi: 10.1016/j.bmc.2009.05.058. Epub 2009 May 29. Bioorg Med Chem. 2009. PMID: 19581099 Free article.

7

1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation.

Biava M, Porretta GC, Poce G, De Logu A, Meleddu R, De Rossi E, Manetti F, Botta M. Biava M, et al. Among authors: de logu a, de rossi e. Eur J Med Chem. 2009 Nov;44(11):4734-8. doi: 10.1016/j.ejmech.2009.06.005. Epub 2009 Jun 13. Eur J Med Chem. 2009. PMID: 19595488

8

Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin.

Biava M, Porretta GC, Poce G, Battilocchio C, Alfonso S, De Logu A, Serra N, Manetti F, Botta M. Biava M, et al. Among authors: de logu a. Bioorg Med Chem. 2010 Nov 15;18(22):8076-84. doi: 10.1016/j.bmc.2010.09.006. Epub 2010 Sep 19. Bioorg Med Chem. 2010. PMID: 20934344

9

Developing pyrrole-derived antimycobacterial agents: a rational lead optimization approach.

Biava M, Porretta GC, Poce G, Battilocchio C, Alfonso S, de Logu A, Manetti F, Botta M. Biava M, et al. Among authors: de logu a. ChemMedChem. 2011 Apr 4;6(4):593-9. doi: 10.1002/cmdc.201000526. Epub 2011 Feb 21. ChemMedChem. 2011. PMID: 21341373 Review.

10

Ungeremine effectively targets mammalian as well as bacterial type I and type II topoisomerases.

Casu L, Cottiglia F, Leonti M, De Logu A, Agus E, Tse-Dinh YC, Lombardo V, Sissi C. Casu L, et al. Among authors: de logu a. Bioorg Med Chem Lett. 2011 Dec 1;21(23):7041-4. doi: 10.1016/j.bmcl.2011.09.097. Epub 2011 Oct 1. Bioorg Med Chem Lett. 2011. PMID: 22014547 Free PMC article.

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