Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
5 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Optimization of 3-(1H-indazol-3-ylmethyl)-1,5-benzodiazepines as potent, orally active CCK-A agonists.
J Med Chem. 1997 Aug 15;40(17):2706-25. doi: 10.1021/jm970265x.
J Med Chem. 1997.
PMID: 9276016
Discovery of 1,5-benzodiazepines with peripheral cholecystokinin (CCK-A) receptor agonist activity (II): Optimization of the C3 amino substituent.
Hirst GC, Aquino C, Birkemo L, Croom DK, Dezube M, Dougherty RW Jr, Ervin GN, Grizzle MK, Henke B, James MK, Johnson MF, Momtahen T, Queen KL, Sherrill RG, Szewczyk J, Willson TM, Sugg EE.
Hirst GC, et al. Among authors: dougherty rw jr.
J Med Chem. 1996 Dec 20;39(26):5236-45. doi: 10.1021/jm9601664.
J Med Chem. 1996.
PMID: 8978852
Item in Clipboard
3-(1H-indazol-3-ylmethyl)-1,5-benzodiazepines: CCK-A agonists that demonstrate oral activity as satiety agents.
Henke BR, Willson TM, Sugg EE, Croom DK, Dougherty RW Jr, Queen KL, Birkemo LS, Ervin GN, Grizzle MK, Johnson MF, James MK.
Henke BR, et al. Among authors: dougherty rw jr.
J Med Chem. 1996 Jul 5;39(14):2655-8. doi: 10.1021/jm960249k.
J Med Chem. 1996.
PMID: 8709093
No abstract available.
Item in Clipboard
Discovery of 1,5-benzodiazepines with peripheral cholecystokinin (CCK-A) receptor agonist activity. 1. Optimization of the agonist "trigger".
Aquino CJ, Armour DR, Berman JM, Birkemo LS, Carr RA, Croom DK, Dezube M, Dougherty RW Jr, Ervin GN, Grizzle MK, Head JE, Hirst GC, James MK, Johnson MF, Miller LJ, Queen KL, Rimele TJ, Smith DN, Sugg EE.
Aquino CJ, et al. Among authors: dougherty rw jr.
J Med Chem. 1996 Jan 19;39(2):562-9. doi: 10.1021/jm950626d.
J Med Chem. 1996.
PMID: 8558528
Item in Clipboard
Modification of receptor selectivity and functional activity in cholecystokinin peptoid ligands.
Dezube M, Sugg EE, Birkemo LS, Croom DK, Dougherty RW Jr, Ervin GN, Grizzle MK, James MK, Johnson MF, Mosher JT, et al.
Dezube M, et al. Among authors: dougherty rw jr.
J Med Chem. 1995 Aug 18;38(17):3384-90. doi: 10.1021/jm00017a022.
J Med Chem. 1995.
PMID: 7650691
Item in Clipboard
Cite
Cite