Durroux T - Search Results

1

Oxytocin and vasopressin agonists and antagonists as research tools and potential therapeutics.

Manning M, Misicka A, Olma A, Bankowski K, Stoev S, Chini B, Durroux T, Mouillac B, Corbani M, Guillon G. Manning M, et al. Among authors: durroux t. J Neuroendocrinol. 2012 Apr;24(4):609-28. doi: 10.1111/j.1365-2826.2012.02303.x. J Neuroendocrinol. 2012. PMID: 22375852 Free PMC article. Review.

2

Design of peptide oxytocin antagonists with strikingly higher affinities and selectivities for the human oxytocin receptor than atosiban.

Manning M, Cheng LL, Stoev S, Wo NC, Chan WY, Szeto HH, Durroux T, Mouillac B, Barberis C. Manning M, et al. Among authors: durroux t. J Pept Sci. 2005 Oct;11(10):593-608. doi: 10.1002/psc.667. J Pept Sci. 2005. PMID: 15880385

3

Peptide and non-peptide agonists and antagonists for the vasopressin and oxytocin V1a, V1b, V2 and OT receptors: research tools and potential therapeutic agents.

Manning M, Stoev S, Chini B, Durroux T, Mouillac B, Guillon G. Manning M, et al. Among authors: durroux t. Prog Brain Res. 2008;170:473-512. doi: 10.1016/S0079-6123(08)00437-8. Prog Brain Res. 2008. PMID: 18655903 Review.

4

Fluorescent agonists and antagonists for vasopressin/oxytocin G protein-coupled receptors: usefulness in ligand screening assays and receptor studies.

Mouillac B, Manning M, Durroux T. Mouillac B, et al. Among authors: durroux t. Mini Rev Med Chem. 2008 Sep;8(10):996-1005. doi: 10.2174/138955708785740607. Mini Rev Med Chem. 2008. PMID: 18782052 Free PMC article. Review.

5

Synthesis and characterization of fluorescent antagonists and agonists for human oxytocin and vasopressin V(1)(a) receptors.

Terrillon S, Cheng LL, Stoev S, Mouillac B, Barberis C, Manning M, Durroux T. Terrillon S, et al. Among authors: durroux t. J Med Chem. 2002 Jun 6;45(12):2579-88. doi: 10.1021/jm010526+. J Med Chem. 2002. PMID: 12036367

6

Conserved aromatic residues in the transmembrane region VI of the V1a vasopressin receptor differentiate agonist vs. antagonist ligand binding.

Cotte N, Balestre MN, Aumelas A, Mahé E, Phalipou S, Morin D, Hibert M, Manning M, Durroux T, Barberis C, Mouillac B. Cotte N, et al. Among authors: durroux t. Eur J Biochem. 2000 Jul;267(13):4253-63. doi: 10.1046/j.1432-1033.2000.01472.x. Eur J Biochem. 2000. PMID: 10866830 Free article.

7

Toward efficient drug screening by homogeneous assays based on the development of new fluorescent vasopressin and oxytocin receptor ligands.

Albizu L, Teppaz G, Seyer R, Bazin H, Ansanay H, Manning M, Mouillac B, Durroux T. Albizu L, et al. Among authors: durroux t. J Med Chem. 2007 Oct 4;50(20):4976-85. doi: 10.1021/jm061404q. Epub 2007 Sep 12. J Med Chem. 2007. PMID: 17850055

8

Subtlety of the structure-affinity and structure-efficacy relationships around a nonpeptide oxytocin receptor agonist.

Frantz MC, Rodrigo J, Boudier L, Durroux T, Mouillac B, Hibert M. Frantz MC, et al. Among authors: durroux t. J Med Chem. 2010 Feb 25;53(4):1546-62. doi: 10.1021/jm901084f. J Med Chem. 2010. PMID: 20104850

9

Time-resolved FRET between GPCR ligands reveals oligomers in native tissues.

Albizu L, Cottet M, Kralikova M, Stoev S, Seyer R, Brabet I, Roux T, Bazin H, Bourrier E, Lamarque L, Breton C, Rives ML, Newman A, Javitch J, Trinquet E, Manning M, Pin JP, Mouillac B, Durroux T. Albizu L, et al. Among authors: durroux t. Nat Chem Biol. 2010 Aug;6(8):587-94. doi: 10.1038/nchembio.396. Epub 2010 Jul 11. Nat Chem Biol. 2010. PMID: 20622858 Free PMC article.

10

Selective fluorescent nonpeptidic antagonists for vasopressin V₂ GPCR: application to ligand screening and oligomerization assays.

Loison S, Cottet M, Orcel H, Adihou H, Rahmeh R, Lamarque L, Trinquet E, Kellenberger E, Hibert M, Durroux T, Mouillac B, Bonnet D. Loison S, et al. Among authors: durroux t. J Med Chem. 2012 Oct 25;55(20):8588-602. doi: 10.1021/jm3006146. Epub 2012 Oct 5. J Med Chem. 2012. PMID: 22984902

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