Inverse agonism at dopamine D2 receptors. Haloperidol-induced prolactin release from GH4C1 cells transfected with the human D2 receptor is antagonized by R(-)-n-propylnorapomorphine, raclopride, and phenoxybenzamine.
Neuropsychopharmacology. 1996 Jul;15(1):53-61. doi: 10.1016/0893-133X(95)00156-8.
Neuropsychopharmacology. 1996.
PMID: 8797192