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Pharmacologic profile of OC000459, a potent, selective, and orally active D prostanoid receptor 2 antagonist that inhibits mast cell-dependent activation of T helper 2 lymphocytes and eosinophils.
Pettipher R, Vinall SL, Xue L, Speight G, Townsend ER, Gazi L, Whelan CJ, Armer RE, Payton MA, Hunter MG. Pettipher R, et al. Among authors: Gazi L. J Pharmacol Exp Ther. 2012 Feb;340(2):473-82. doi: 10.1124/jpet.111.187203. Epub 2011 Nov 21. J Pharmacol Exp Ther. 2012. PMID: 22106101
Delta12-prostaglandin D2 is a potent and selective CRTH2 receptor agonist and causes activation of human eosinophils and Th2 lymphocytes.
Gazi L, Gyles S, Rose J, Lees S, Allan C, Xue L, Jassal R, Speight G, Gamble V, Pettipher R. Gazi L, et al. Prostaglandins Other Lipid Mediat. 2005 Jan;75(1-4):153-67. doi: 10.1016/j.prostaglandins.2004.11.003. Prostaglandins Other Lipid Mediat. 2005. PMID: 15789622
Indole-3-acetic acid antagonists of the prostaglandin D2 receptor CRTH2.
Armer RE, Ashton MR, Boyd EA, Brennan CJ, Brookfield FA, Gazi L, Gyles SL, Hay PA, Hunter MG, Middlemiss D, Whittaker M, Xue L, Pettipher R. Armer RE, et al. Among authors: Gazi L. J Med Chem. 2005 Oct 6;48(20):6174-7. doi: 10.1021/jm050519b. J Med Chem. 2005. PMID: 16190744
Constitutive oligomerization of human D2 dopamine receptors expressed in Spodoptera frugiperda 9 (Sf9) and in HEK293 cells. Analysis using co-immunoprecipitation and time-resolved fluorescence resonance energy transfer.
Gazi L, López-Giménez JF, Rüdiger MP, Strange PG. Gazi L, et al. Eur J Biochem. 2003 Oct;270(19):3928-38. doi: 10.1046/j.1432-1033.2003.03773.x. Eur J Biochem. 2003. PMID: 14511374 Free article.
The agonist activities of the putative antipsychotic agents, L-745,870 and U-101958 in HEK293 cells expressing the human dopamine D4.4 receptor.
Gazi L, Bobirnac I, Danzeisen M, Schüpbach E, Bruinvels AT, Geisse S, Sommer B, Hoyer D, Tricklebank M, Schoeffter P. Gazi L, et al. Br J Pharmacol. 1998 Jul;124(5):889-96. doi: 10.1038/sj.bjp.0701921. Br J Pharmacol. 1998. PMID: 9692773 Free PMC article.
L-745,870 and U-101958 also inhibited forskolin-stimulated cyclic AMP accumulation in HEK293/D4 cells in a concentration-dependent way. L-745,870 was less efficacious than dopamine (71% the efficacy of dopamine), whereas U-101958 behaved as a full agonist compared to dopamine. ...
L-745,870 and U-101958 also inhibited forskolin-stimulated cyclic AMP accumulation in HEK293/D4 cells in a concentration-dependent wa
Formation of oligomers by G protein-coupled receptors.
Gazi L, López-Giménez JF, Strange PG. Gazi L, et al. Curr Opin Drug Discov Devel. 2002 Sep;5(5):756-63. Curr Opin Drug Discov Devel. 2002. PMID: 12630296 Review.
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