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Breakpoint analysis of transcriptional and genomic profiles uncovers novel gene fusions spanning multiple human cancer types.
PLoS Genet. 2013 Apr;9(4):e1003464. doi: 10.1371/journal.pgen.1003464. Epub 2013 Apr 25.
PLoS Genet. 2013.
PMID: 23637631
Free PMC article.
PharmGKB summary: sorafenib pathways.
Gong L, Giacomini MM, Giacomini C, Maitland ML, Altman RB, Klein TE.
Gong L, et al. Among authors: giacomini mm.
Pharmacogenet Genomics. 2017 Jun;27(6):240-246. doi: 10.1097/FPC.0000000000000279.
Pharmacogenet Genomics. 2017.
PMID: 28362716
Free PMC article.
Review.
No abstract available.
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Epithelial cells utilize cortical actin/myosin to activate latent TGF-β through integrin α(v)β(6)-dependent physical force.
Giacomini MM, Travis MA, Kudo M, Sheppard D.
Giacomini MM, et al.
Exp Cell Res. 2012 Apr 1;318(6):716-22. doi: 10.1016/j.yexcr.2012.01.020. Epub 2012 Jan 28.
Exp Cell Res. 2012.
PMID: 22309779
Free PMC article.
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Metformin Is a Substrate and Inhibitor of the Human Thiamine Transporter, THTR-2 (SLC19A3).
Liang X, Chien HC, Yee SW, Giacomini MM, Chen EC, Piao M, Hao J, Twelves J, Lepist EI, Ray AS, Giacomini KM.
Liang X, et al. Among authors: giacomini mm.
Mol Pharm. 2015 Dec 7;12(12):4301-10. doi: 10.1021/acs.molpharmaceut.5b00501. Epub 2015 Nov 16.
Mol Pharm. 2015.
PMID: 26528626
Free PMC article.
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Targeting of αv integrin identifies a core molecular pathway that regulates fibrosis in several organs.
Henderson NC, Arnold TD, Katamura Y, Giacomini MM, Rodriguez JD, McCarty JH, Pellicoro A, Raschperger E, Betsholtz C, Ruminski PG, Griggs DW, Prinsen MJ, Maher JJ, Iredale JP, Lacy-Hulbert A, Adams RH, Sheppard D.
Henderson NC, et al. Among authors: giacomini mm.
Nat Med. 2013 Dec;19(12):1617-24. doi: 10.1038/nm.3282. Epub 2013 Nov 10.
Nat Med. 2013.
PMID: 24216753
Free PMC article.
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Metabolomic and Genome-wide Association Studies Reveal Potential Endogenous Biomarkers for OATP1B1.
Yee SW, Giacomini MM, Hsueh CH, Weitz D, Liang X, Goswami S, Kinchen JM, Coelho A, Zur AA, Mertsch K, Brian W, Kroetz DL, Giacomini KM.
Yee SW, et al. Among authors: giacomini mm.
Clin Pharmacol Ther. 2016 Nov;100(5):524-536. doi: 10.1002/cpt.434. Epub 2016 Sep 20.
Clin Pharmacol Ther. 2016.
PMID: 27447836
Free PMC article.
Clinical Trial.
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Organic Anion Transporter Polypeptide 1B1 Polymorphism Modulates the Extent of Drug-Drug Interaction and Associated Biomarker Levels in Healthy Volunteers.
Yee SW, Giacomini MM, Shen H, Humphreys WG, Horng H, Brian W, Lai Y, Kroetz DL, Giacomini KM.
Yee SW, et al. Among authors: giacomini mm.
Clin Transl Sci. 2019 Jul;12(4):388-399. doi: 10.1111/cts.12625. Epub 2019 Apr 13.
Clin Transl Sci. 2019.
PMID: 30982223
Free PMC article.
Clinical Trial.
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Interaction of 2,4-Diaminopyrimidine-Containing Drugs Including Fedratinib and Trimethoprim with Thiamine Transporters.
Giacomini MM, Hao J, Liang X, Chandrasekhar J, Twelves J, Whitney JA, Lepist EI, Ray AS.
Giacomini MM, et al.
Drug Metab Dispos. 2017 Jan;45(1):76-85. doi: 10.1124/dmd.116.073338. Epub 2016 Nov 1.
Drug Metab Dispos. 2017.
PMID: 27803021
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