Goins CM - Search Results

1

Structure-Based Optimization of ML300-Derived, Noncovalent Inhibitors Targeting the Severe Acute Respiratory Syndrome Coronavirus 3CL Protease (SARS-CoV-2 3CL^pro).

Han SH, Goins CM, Arya T, Shin WJ, Maw J, Hooper A, Sonawane DP, Porter MR, Bannister BE, Crouch RD, Lindsey AA, Lakatos G, Martinez SR, Alvarado J, Akers WS, Wang NS, Jung JU, Macdonald JD, Stauffer SR. Han SH, et al. Among authors: goins cm. J Med Chem. 2022 Feb 24;65(4):2880-2904. doi: 10.1021/acs.jmedchem.1c00598. Epub 2021 Aug 4. J Med Chem. 2022. PMID: 34347470 Free PMC article.

2

Hexose-6-phosphate dehydrogenase blockade reverses prostate cancer drug resistance in xenograft models by glucocorticoid inactivation.

Li J, Berk M, Alyamani M, Sabharwal N, Goins C, Alvarado J, Baratchian M, Zhu Z, Stauffer S, Klein EA, Sharifi N. Li J, et al. Sci Transl Med. 2021 May 26;13(595):eabe8226. doi: 10.1126/scitranslmed.abe8226. Sci Transl Med. 2021. PMID: 34039740 Free PMC article.

3

Discovery and Characterization of Selective, First-in-Class Inhibitors of Citron Kinase.

Maw JJ, Coker JA, Arya T, Goins CM, Sonawane D, Han SH, Rees MG, Ronan MM, Roth JA, Wang NS, Heemers HV, Macdonald JD, Stauffer SR. Maw JJ, et al. Among authors: goins cm. J Med Chem. 2024 Feb 22;67(4):2631-2666. doi: 10.1021/acs.jmedchem.3c01807. Epub 2024 Feb 8. J Med Chem. 2024. PMID: 38330278

4

Structural basis for lipid binding and mechanism of the Mycobacterium tuberculosis Rv3802 phospholipase.

Goins CM, Schreidah CM, Dajnowicz S, Ronning DR. Goins CM, et al. J Biol Chem. 2018 Jan 26;293(4):1363-1372. doi: 10.1074/jbc.RA117.000240. Epub 2017 Dec 15. J Biol Chem. 2018. PMID: 29247008 Free PMC article.

5

Mycolyltransferase from Mycobacterium tuberculosis in covalent complex with tetrahydrolipstatin provides insights into antigen 85 catalysis.

Goins CM, Dajnowicz S, Smith MD, Parks JM, Ronning DR. Goins CM, et al. J Biol Chem. 2018 Mar 9;293(10):3651-3662. doi: 10.1074/jbc.RA117.001681. Epub 2018 Jan 19. J Biol Chem. 2018. PMID: 29352107 Free PMC article.

6

Thermal and Photoinduced Copper-Promoted C-Se Bond Formation: Synthesis of 2-Alkyl-1,2-benzisoselenazol-3(2H)-ones and Evaluation against Mycobacterium tuberculosis.

Thanna S, Goins CM, Knudson SE, Slayden RA, Ronning DR, Sucheck SJ. Thanna S, et al. Among authors: goins cm. J Org Chem. 2017 Apr 7;82(7):3844-3854. doi: 10.1021/acs.joc.7b00440. Epub 2017 Mar 20. J Org Chem. 2017. PMID: 28273423 Free PMC article.

7

Synthesis and evaluation of new 2-aminothiophenes against Mycobacterium tuberculosis.

Thanna S, Knudson SE, Grzegorzewicz A, Kapil S, Goins CM, Ronning DR, Jackson M, Slayden RA, Sucheck SJ. Thanna S, et al. Among authors: goins cm. Org Biomol Chem. 2016 Jul 7;14(25):6119-6133. doi: 10.1039/c6ob00821f. Epub 2016 Jun 2. Org Biomol Chem. 2016. PMID: 27251120 Free PMC article.

8

Exploring Covalent Allosteric Inhibition of Antigen 85C from Mycobacterium tuberculosis by Ebselen Derivatives.

Goins CM, Dajnowicz S, Thanna S, Sucheck SJ, Parks JM, Ronning DR. Goins CM, et al. ACS Infect Dis. 2017 May 12;3(5):378-387. doi: 10.1021/acsinfecdis.7b00003. Epub 2017 Mar 21. ACS Infect Dis. 2017. PMID: 28285521 Free PMC article.

9

Characterization of Tetrahydrolipstatin and Stereoderivatives on the Inhibition of Essential Mycobacterium tuberculosis Lipid Esterases.

Goins CM, Sudasinghe TD, Liu X, Wang Y, O'Doherty GA, Ronning DR. Goins CM, et al. Biochemistry. 2018 Apr 24;57(16):2383-2393. doi: 10.1021/acs.biochem.8b00152. Epub 2018 Apr 10. Biochemistry. 2018. PMID: 29601187 Free PMC article.

10

Biochemical and microbiological evaluation of N-aryl urea derivatives against mycobacteria and mycobacterial hydrolases.

Vartak A, Goins C, de Moura VCN, Schreidah CM, Landgraf AD, Lin B, Du J, Jackson M, Ronning DR, Sucheck SJ. Vartak A, et al. Among authors: goins c. Medchemcomm. 2019 Jun 4;10(7):1197-1204. doi: 10.1039/c9md00122k. eCollection 2019 Jul 1. Medchemcomm. 2019. PMID: 31741730 Free PMC article.

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