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Discovery of 4-((2S,4S)-4-Ethoxy-1-((5-methoxy-7-methyl-1H-indol-4-yl)methyl)piperidin-2-yl)benzoic Acid (LNP023), a Factor B Inhibitor Specifically Designed To Be Applicable to Treating a Diverse Array of Complement Mediated Diseases.
J Med Chem. 2020 Jun 11;63(11):5697-5722. doi: 10.1021/acs.jmedchem.9b01870. Epub 2020 Feb 19.
J Med Chem. 2020.
PMID: 32073845
Design, Synthesis, and Preclinical Characterization of Selective Factor D Inhibitors Targeting the Alternative Complement Pathway.
Karki RG, Powers J, Mainolfi N, Anderson K, Belanger DB, Liu D, Ji N, Jendza K, Gelin CF, Mac Sweeney A, Solovay C, Delgado O, Crowley M, Liao SM, Argikar UA, Flohr S, La Bonte LR, Lorthiois EL, Vulpetti A, Brown A, Long D, Prentiss M, Gradoux N, de Erkenez A, Cumin F, Adams C, Jaffee B, Mogi M.
Karki RG, et al. Among authors: gradoux n.
J Med Chem. 2019 May 9;62(9):4656-4668. doi: 10.1021/acs.jmedchem.9b00271. Epub 2019 Apr 30.
J Med Chem. 2019.
PMID: 30995036
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Fluorescence Lifetime-Based Competitive Binding Assays for Measuring the Binding Potency of Protease Inhibitors In Vitro.
Boettcher A, Gradoux N, Lorthiois E, Brandl T, Orain D, Schiering N, Cumin F, Woelcke J, Hassiepen U.
Boettcher A, et al. Among authors: gradoux n.
J Biomol Screen. 2014 Jul;19(6):870-7. doi: 10.1177/1087057114521295. Epub 2014 Jan 31.
J Biomol Screen. 2014.
PMID: 24487225
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Effects of intestinal fatty acid-binding protein overexpression on fatty acid metabolism in Caco-2 cells.
Darimont C, Gradoux N, Persohn E, Cumin F, De Pover A.
Darimont C, et al. Among authors: gradoux n.
J Lipid Res. 2000 Jan;41(1):84-92.
J Lipid Res. 2000.
PMID: 10627505
Free article.
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Differential regulation of intestinal and liver fatty acid-binding proteins in human intestinal cell line (Caco-2): role of collagen.
Darimont C, Gradoux N, Cumin F, Baum HP, De Pover A.
Darimont C, et al. Among authors: gradoux n.
Exp Cell Res. 1998 Nov 1;244(2):441-7. doi: 10.1006/excr.1998.4186.
Exp Cell Res. 1998.
PMID: 9806794
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Characterisation of Na/K-ATPase, its isoforms, and the inotropic response to ouabain in isolated failing human hearts.
Shamraj OI, Grupp IL, Grupp G, Melvin D, Gradoux N, Kremers W, Lingrel JB, De Pover A.
Shamraj OI, et al. Among authors: gradoux n.
Cardiovasc Res. 1993 Dec;27(12):2229-37. doi: 10.1093/cvr/27.12.2229.
Cardiovasc Res. 1993.
PMID: 8313433
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Epidermal growth factor regulates fatty acid uptake and metabolism in Caco-2 cells.
Darimont C, Gradoux N, de Pover A.
Darimont C, et al. Among authors: gradoux n.
Am J Physiol. 1999 Mar;276(3):G606-12. doi: 10.1152/ajpgi.1999.276.3.G606.
Am J Physiol. 1999.
PMID: 10070036
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