Hübner H - Search Results

1

Synthesis, biological evaluation and radiolabelling by 18F-fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET.

Höfling SB, Maschauer S, Hübner H, Gmeiner P, Wester HJ, Prante O, Heinrich MR. Höfling SB, et al. Among authors: hubner h. Bioorg Med Chem Lett. 2010 Dec 1;20(23):6933-7. doi: 10.1016/j.bmcl.2010.09.142. Epub 2010 Oct 26. Bioorg Med Chem Lett. 2010. PMID: 21030255

2

Azaindole derivatives with high affinity for the dopamine D4 receptor: synthesis, ligand binding studies and comparison of molecular electrostatic potential maps.

Löber S, Hübner H, Gmeiner P. Löber S, et al. Among authors: hubner h. Bioorg Med Chem Lett. 1999 Jan 4;9(1):97-102. doi: 10.1016/s0960-894x(98)00692-1. Bioorg Med Chem Lett. 1999. PMID: 9990464

3

Enantio- and diastereocontrolled dopamine D1, D2, D3 and D4 receptor binding of N-(3-pyrrolidinylmethyl)benzamides synthesized from aspartic acid.

Thomas C, Hübner H, Gmeiner P. Thomas C, et al. Among authors: hubner h. Bioorg Med Chem Lett. 1999 Mar 22;9(6):841-6. doi: 10.1016/s0960-894x(99)00086-4. Bioorg Med Chem Lett. 1999. PMID: 10206547

4

2,2-Dicyanovinyl as a nonaromatic aryl bioisostere: synthesis, binding experiments and SAR studies of highly selective dopamine D4 receptor ligands.

Haubmann C, Hübner H, Gmeiner P. Haubmann C, et al. Among authors: hubner h. Bioorg Med Chem Lett. 1999 Jul 19;9(14):1969-72. doi: 10.1016/s0960-894x(99)00302-9. Bioorg Med Chem Lett. 1999. PMID: 10450964

5

Piperidinylpyrroles: design, synthesis and binding properties of novel and selective dopamine D4 receptor ligands.

Haubmann C, Hübner H, Gmeiner P. Haubmann C, et al. Among authors: hubner h. Bioorg Med Chem Lett. 1999 Nov 1;9(21):3143-6. doi: 10.1016/s0960-894x(99)00540-5. Bioorg Med Chem Lett. 1999. PMID: 10560741

6

Conjugated enynes as nonaromatic catechol bioisosteres: synthesis, binding experiments, and computational studies of novel dopamine receptor agonists recognizing preferentially the D(3) subtype.

Hübner H, Haubmann C, Utz W, Gmeiner P. Hübner H, et al. J Med Chem. 2000 Feb 24;43(4):756-62. doi: 10.1021/jm991098z. J Med Chem. 2000. PMID: 10691700

7

Phenyloxazoles and phenylthiazoles as benzamide bioisosteres: synthesis and dopamine receptor binding profiles.

Einsiedel J, Thomas C, Hübner H, Gmeiner P. Einsiedel J, et al. Among authors: hubner h. Bioorg Med Chem Lett. 2000 Sep 4;10(17):2041-4. doi: 10.1016/s0960-894x(00)00405-4. Bioorg Med Chem Lett. 2000. PMID: 10987445

8

Azepino- and diazepinoindoles: synthesis and dopamine receptor binding profiles.

Kraxner J, Hübner H, Gmeiner P. Kraxner J, et al. Among authors: hubner h. Arch Pharm (Weinheim). 2000 Sep;333(9):287-92. doi: 10.1002/1521-4184(20009)333:9<287::aid-ardp287>3.0.co;2-r. Arch Pharm (Weinheim). 2000. PMID: 11039184

9

Cyanoindole derivatives as highly selective dopamine D(4) receptor partial agonists: solid-phase synthesis, binding assays, and functional experiments.

Hübner H, Kraxner J, Gmeiner P. Hübner H, et al. J Med Chem. 2000 Nov 16;43(23):4563-9. doi: 10.1021/jm0009989. J Med Chem. 2000. PMID: 11087581

10

Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213).

Löber S, Hübner H, Utz W, Gmeiner P. Löber S, et al. Among authors: hubner h. J Med Chem. 2001 Aug 16;44(17):2691-4. doi: 10.1021/jm015522j. J Med Chem. 2001. PMID: 11495580

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