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6,656 results
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Identification of a dual δ OR antagonist/μ OR agonist as a potential therapeutic for diarrhea-predominant Irritable Bowel Syndrome (IBS-d).
Breslin HJ, Diamond CJ, Kavash RW, Cai C, Dyatkin AB, Miskowski TA, Zhang SP, Wade PR, Hornby PJ, He W. Breslin HJ, et al. Bioorg Med Chem Lett. 2012 Jul 15;22(14):4869-72. doi: 10.1016/j.bmcl.2012.05.042. Epub 2012 May 24. Bioorg Med Chem Lett. 2012. PMID: 22695132
Aza-bicyclic amino acid sulfonamides as alpha(4)beta(1)/alpha(4)beta(7) integrin antagonists.
Dyatkin AB, Hoekstra WJ, Kinney WA, Kontoyianni M, Santulli RJ, Kimball ES, Fisher MC, Prouty SM, Abraham WM, de Garavilla L, Andrade-Gordon P, Hlasta DJ, He W, Hornby PJ, Damiano BP, Maryanoff BE. Dyatkin AB, et al. Bioorg Med Chem Lett. 2004 Feb 9;14(3):591-6. doi: 10.1016/j.bmcl.2003.11.063. Bioorg Med Chem Lett. 2004. PMID: 14741249
Stimulation of cortical bone formation with thienopyrimidine based inhibitors of Notum Pectinacetylesterase.
Tarver JE Jr, Pabba PK, Barbosa J, Han Q, Gardyan MW, Brommage R, Thompson AY, Schmidt JM, Wilson AGE, He W, Lombardo VK, Carson KG. Tarver JE Jr, et al. Bioorg Med Chem Lett. 2016 Mar 15;26(6):1525-1528. doi: 10.1016/j.bmcl.2016.02.021. Epub 2016 Feb 10. Bioorg Med Chem Lett. 2016. PMID: 26897593
A novel protocol to accelerate dynamic combinatorial chemistry via isolation of ligand-target adducts from dynamic combinatorial libraries: a case study identifying competitive inhibitors of lysozyme.
Fang Z, He W, Li X, Li Z, Chen B, Ouyang P, Guo K. Fang Z, et al. Bioorg Med Chem Lett. 2013 Sep 15;23(18):5174-7. doi: 10.1016/j.bmcl.2013.07.011. Epub 2013 Jul 17. Bioorg Med Chem Lett. 2013. PMID: 23932789
Spirocyclic ureas: orally bioavailable 11 beta-HSD1 inhibitors identified by computer-aided drug design.
Tice CM, Zhao W, Xu Z, Cacatian ST, Simpson RD, Ye YJ, Singh SB, McKeever BM, Lindblom P, Guo J, Krosky PM, Kruk BA, Berbaum J, Harrison RK, Johnson JJ, Bukhtiyarov Y, Panemangalore R, Scott BB, Zhao Y, Bruno JG, Zhuang L, McGeehan GM, He W, Claremon DA. Tice CM, et al. Bioorg Med Chem Lett. 2010 Feb 1;20(3):881-6. doi: 10.1016/j.bmcl.2009.12.082. Epub 2010 Jan 4. Bioorg Med Chem Lett. 2010. PMID: 20064717
Triazinediones as prokineticin 1 receptor antagonists. Part 1: SAR, synthesis and biological evaluation.
Ralbovsky JL, Lisko JG, Palmer JM, Mabus J, Chevalier KM, Schulz MJ, Dyatkin AB, Miskowski TA, Coats SJ, Hornby P, He W. Ralbovsky JL, et al. Bioorg Med Chem Lett. 2009 May 15;19(10):2661-3. doi: 10.1016/j.bmcl.2009.03.157. Epub 2009 Apr 5. Bioorg Med Chem Lett. 2009. PMID: 19375913
Design and optimization of aniline-substituted tetrahydroquinoline C5a receptor antagonists.
Gong Y, Barbay JK, Buntinx M, Li J, Wauwe JV, Claes C, Lommen GV, Hornby PJ, He W. Gong Y, et al. Bioorg Med Chem Lett. 2008 Jul 15;18(14):3852-5. doi: 10.1016/j.bmcl.2008.06.059. Epub 2008 Jun 20. Bioorg Med Chem Lett. 2008. PMID: 18595693
Synthesis and characterization of 5,6,7,8-tetrahydroquinoline C5a receptor antagonists.
Barbay JK, Gong Y, Buntinx M, Li J, Claes C, Hornby PJ, Van Lommen G, Van Wauwe J, He W. Barbay JK, et al. Bioorg Med Chem Lett. 2008 Apr 15;18(8):2544-8. doi: 10.1016/j.bmcl.2008.03.049. Epub 2008 Mar 20. Bioorg Med Chem Lett. 2008. PMID: 18378452
Synthesis and SAR of pyridazinone-substituted phenylalanine amide alpha4 integrin antagonists.
Gong Y, Kent Barbay J, Kimball ES, Santulli RJ, Carolyn Fisher M, Dyatkin AB, Miskowski TA, Hornby PJ, He W. Gong Y, et al. Bioorg Med Chem Lett. 2008 Feb 15;18(4):1331-5. doi: 10.1016/j.bmcl.2008.01.022. Epub 2008 Jan 11. Bioorg Med Chem Lett. 2008. PMID: 18226905
Synthesis and biological evaluation of novel pyridazinone-based alpha4 integrin receptor antagonists.
Gong Y, Barbay JK, Dyatkin AB, Miskowski TA, Kimball ES, Prouty SM, Fisher MC, Santulli RJ, Schneider CR, Wallace NH, Ballentine SA, Hageman WE, Masucci JA, Maryanoff BE, Damiano BP, Andrade-Gordon P, Hlasta DJ, Hornby PJ, He W. Gong Y, et al. J Med Chem. 2006 Jun 1;49(11):3402-11. doi: 10.1021/jm060031q. J Med Chem. 2006. PMID: 16722660
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