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Design of Conformationally Constrained Acyl Sulfonamide Isosteres: Identification of N-([1,2,4]Triazolo[4,3- a]pyridin-3-yl)methane-sulfonamides as Potent and Selective hNaV1.7 Inhibitors for the Treatment of Pain.
J Med Chem. 2018 Jun 14;61(11):4810-4831. doi: 10.1021/acs.jmedchem.7b01826. Epub 2018 May 23.
J Med Chem. 2018.
PMID: 29737846
Discovery of Aryl Sulfonamides as Isoform-Selective Inhibitors of NaV1.7 with Efficacy in Rodent Pain Models.
Focken T, Liu S, Chahal N, Dauphinais M, Grimwood ME, Chowdhury S, Hemeon I, Bichler P, Bogucki D, Waldbrook M, Bankar G, Sojo LE, Young C, Lin S, Shuart N, Kwan R, Pang J, Chang JH, Safina BS, Sutherlin DP, Johnson JP Jr, Dehnhardt CM, Mansour TS, Oballa RM, Cohen CJ, Robinette CL.
Focken T, et al. Among authors: hemeon i.
ACS Med Chem Lett. 2016 Jan 19;7(3):277-82. doi: 10.1021/acsmedchemlett.5b00447. eCollection 2016 Mar 10.
ACS Med Chem Lett. 2016.
PMID: 26985315
Free PMC article.
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Identification of Selective Acyl Sulfonamide-Cycloalkylether Inhibitors of the Voltage-Gated Sodium Channel (NaV) 1.7 with Potent Analgesic Activity.
Sun S, Jia Q, Zenova AY, Wilson MS, Chowdhury S, Focken T, Li J, Decker S, Grimwood ME, Andrez JC, Hemeon I, Sheng T, Chen CA, White A, Hackos DH, Deng L, Bankar G, Khakh K, Chang E, Kwan R, Lin S, Nelkenbrecher K, Sellers BD, DiPasquale AG, Chang J, Pang J, Sojo L, Lindgren A, Waldbrook M, Xie Z, Young C, Johnson JP, Robinette CL, Cohen CJ, Safina BS, Sutherlin DP, Ortwine DF, Dehnhardt CM.
Sun S, et al. Among authors: hemeon i.
J Med Chem. 2019 Jan 24;62(2):908-927. doi: 10.1021/acs.jmedchem.8b01621. Epub 2018 Dec 21.
J Med Chem. 2019.
PMID: 30499663
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Discovery of Acyl-sulfonamide Nav1.7 Inhibitors GDC-0276 and GDC-0310.
Safina BS, McKerrall SJ, Sun S, Chen CA, Chowdhury S, Jia Q, Li J, Zenova AY, Andrez JC, Bankar G, Bergeron P, Chang JH, Chang E, Chen J, Dean R, Decker SM, DiPasquale A, Focken T, Hemeon I, Khakh K, Kim A, Kwan R, Lindgren A, Lin S, Maher J, Mezeyova J, Misner D, Nelkenbrecher K, Pang J, Reese R, Shields SD, Sojo L, Sheng T, Verschoof H, Waldbrook M, Wilson MS, Xie Z, Young C, Zabka TS, Hackos DH, Ortwine DF, White AD, Johnson JP Jr, Robinette CL, Dehnhardt CM, Cohen CJ, Sutherlin DP.
Safina BS, et al. Among authors: hemeon i.
J Med Chem. 2021 Mar 25;64(6):2953-2966. doi: 10.1021/acs.jmedchem.1c00049. Epub 2021 Mar 8.
J Med Chem. 2021.
PMID: 33682420
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Synthesis of 4-deoxy-4-nitrosialic acid.
Hemeon I, Bennet AJ.
Hemeon I, et al.
Org Biomol Chem. 2006 Aug 7;4(15):2986-92. doi: 10.1039/b605218e. Epub 2006 Jul 5.
Org Biomol Chem. 2006.
PMID: 16855749
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Characterizing DNA methyltransferases with an ultrasensitive luciferase-linked continuous assay.
Hemeon I, Gutierrez JA, Ho MC, Schramm VL.
Hemeon I, et al.
Anal Chem. 2011 Jun 15;83(12):4996-5004. doi: 10.1021/ac200816m. Epub 2011 May 16.
Anal Chem. 2011.
PMID: 21545095
Free PMC article.
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Growth and metastases of human lung cancer are inhibited in mouse xenografts by a transition state analogue of 5'-methylthioadenosine phosphorylase.
Basu I, Locker J, Cassera MB, Belbin TJ, Merino EF, Dong X, Hemeon I, Evans GB, Guha C, Schramm VL.
Basu I, et al. Among authors: hemeon i.
J Biol Chem. 2011 Feb 11;286(6):4902-11. doi: 10.1074/jbc.M110.198374. Epub 2010 Dec 6.
J Biol Chem. 2011.
PMID: 21135097
Free PMC article.
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Silylstannation of terminal alkynes using a recyclable palladium(0) catalyst immobilised in an ionic liquid.
Hemeon I, Singer RD.
Hemeon I, et al.
Chem Commun (Camb). 2002 Sep 7;(17):1884-5. doi: 10.1039/b205999a.
Chem Commun (Camb). 2002.
PMID: 12271657
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