Janssens F - Search Results

1

Selection of a respiratory syncytial virus fusion inhibitor clinical candidate. 2. Discovery of a morpholinopropylaminobenzimidazole derivative (TMC353121).

Bonfanti JF, Meyer C, Doublet F, Fortin J, Muller P, Queguiner L, Gevers T, Janssens P, Szel H, Willebrords R, Timmerman P, Wuyts K, van Remoortere P, Janssens F, Wigerinck P, Andries K. Bonfanti JF, et al. Among authors: janssens p, janssens f. J Med Chem. 2008 Feb 28;51(4):875-96. doi: 10.1021/jm701284j. Epub 2008 Feb 7. J Med Chem. 2008. PMID: 18254606

2

Selection of a respiratory syncytial virus fusion inhibitor clinical candidate, part 1: improving the pharmacokinetic profile using the structure-property relationship.

Bonfanti JF, Doublet F, Fortin J, Lacrampe J, Guillemont J, Muller P, Queguiner L, Arnoult E, Gevers T, Janssens P, Szel H, Willebrords R, Timmerman P, Wuyts K, Janssens F, Sommen C, Wigerinck P, Andries K. Bonfanti JF, et al. Among authors: janssens p, janssens f. J Med Chem. 2007 Sep 20;50(19):4572-84. doi: 10.1021/jm070143x. Epub 2007 Aug 28. J Med Chem. 2007. PMID: 17722899

3

Substituted benzimidazoles with nanomolar activity against respiratory syncytial virus.

Andries K, Moeremans M, Gevers T, Willebrords R, Sommen C, Lacrampe J, Janssens F, Wyde PR. Andries K, et al. Among authors: janssens f. Antiviral Res. 2003 Nov;60(3):209-19. doi: 10.1016/j.antiviral.2003.07.004. Antiviral Res. 2003. PMID: 14638397

4

Norpiperidine imidazoazepines as a new class of potent, selective, and nonsedative H1 antihistamines.

Janssens F, Leenaerts J, Diels G, De Boeck B, Megens A, Langlois X, van Rossem K, Beetens J, Borgers M. Janssens F, et al. J Med Chem. 2005 Mar 24;48(6):2154-66. doi: 10.1021/jm049495j. J Med Chem. 2005. PMID: 15771458

5

4-Phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives, a novel class of selective delta-opioid agonists.

Trabanco AA, Pullan S, Alonso JM, Alvarez RM, Andrés JI, Boeckx I, Fernández J, Gómez A, Iturrino L, Janssens FE, Leenaerts JE, De Lucas AI, Matesanz E, Meert T, Steckler T. Trabanco AA, et al. Bioorg Med Chem Lett. 2006 Jan 1;16(1):146-9. doi: 10.1016/j.bmcl.2005.09.025. Epub 2005 Oct 19. Bioorg Med Chem Lett. 2006. PMID: 16236510

6

4-Phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives as non-peptidic selective delta-opioid agonists with potential anxiolytic/antidepressant properties. Part 2.

Trabanco AA, Aerts N, Alvarez RM, Andrés JI, Boeckx I, Fernández J, Gómez A, Janssens FE, Leenaerts JE, De Lucas AI, Matesanz E, Steckler T, Pullan S. Trabanco AA, et al. Bioorg Med Chem Lett. 2007 Jul 15;17(14):3860-3. doi: 10.1016/j.bmcl.2007.05.012. Epub 2007 May 10. Bioorg Med Chem Lett. 2007. PMID: 17512730

7

Synthetic 1,4-disubstituted-1,4-dihydro-5H-tetrazol-5-one derivatives of fentanyl: alfentanil (R 39209), a potent, extremely short-acting narcotic analgesic.

Janssens F, Torremans J, Janssen PA. Janssens F, et al. J Med Chem. 1986 Nov;29(11):2290-7. doi: 10.1021/jm00161a027. J Med Chem. 1986. PMID: 2878076

8

New antihistaminic N-heterocyclic 4-piperidinamines. 1. Synthesis and antihistaminic activity of N-(4-piperidinyl)-1H-benzimidazol-2-amines.

Janssens F, Torremans J, Janssen M, Stokbroekx RA, Luyckx M, Janssen PA. Janssens F, et al. J Med Chem. 1985 Dec;28(12):1925-33. doi: 10.1021/jm00150a028. J Med Chem. 1985. PMID: 4068010

9

New antihistaminic N-heterocyclic 4-piperidinamines. 2. Synthesis and antihistaminic activity of 1-[(4-fluorophenyl)methyl]-N-(4-piperidinyl)-1H-benzimidazol-2-a mines.

Janssens F, Torremans J, Janssen M, Stokbroekx RA, Luyckx M, Janssen PA. Janssens F, et al. J Med Chem. 1985 Dec;28(12):1934-43. doi: 10.1021/jm00150a029. J Med Chem. 1985. PMID: 3934386

10

New antihistaminic N-heterocyclic 4-piperidinamines. 3. Synthesis and antihistaminic activity of N-(4-piperidinyl)-3H-imidazo[4,5-b]pyridin-2-amines.

Janssens F, Torremans J, Janssen M, Stokbroekx RA, Luyckx M, Janssen PA. Janssens F, et al. J Med Chem. 1985 Dec;28(12):1943-7. doi: 10.1021/jm00150a030. J Med Chem. 1985. PMID: 3934387

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