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Functional characterization of Tet-AMPA [tetrazolyl-2-amino-3-(3-hydroxy-5-methyl- 4-isoxazolyl)propionic acid] analogues at ionotropic glutamate receptors GluR1-GluR4. The molecular basis for the functional selectivity profile of 2-Bn-Tet-AMPA.
Jensen AA, Christesen T, Bølcho U, Greenwood JR, Postorino G, Vogensen SB, Johansen TN, Egebjerg J, Bräuner-Osborne H, Clausen RP. Jensen AA, et al. Among authors: johansen tn. J Med Chem. 2007 Aug 23;50(17):4177-85. doi: 10.1021/jm070532r. Epub 2007 Aug 2. J Med Chem. 2007. PMID: 17672447
Pharmacological characterization and binding modes of novel racemic and optically active phenylalanine-based antagonists of AMPA receptors.
Szymańska E, Nielsen B, Johansen TN, Cuñado Moral AM, Pickering DS, Szczepańska K, Mickowska A, Kieć-Kononowicz K. Szymańska E, et al. Among authors: johansen tn. Eur J Med Chem. 2017 Sep 29;138:874-883. doi: 10.1016/j.ejmech.2017.07.007. Epub 2017 Jul 8. Eur J Med Chem. 2017. PMID: 28738307
Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands.
Szymańska E, Chałupnik P, Szczepańska K, Cuñado Moral AM, Pickering DS, Nielsen B, Johansen TN, Kieć-Kononowicz K. Szymańska E, et al. Among authors: johansen tn. Bioorg Med Chem Lett. 2016 Nov 15;26(22):5568-5572. doi: 10.1016/j.bmcl.2016.09.075. Epub 2016 Sep 30. Bioorg Med Chem Lett. 2016. PMID: 27765511
4-hydroxy-1,2,5-oxadiazol-3-yl moiety as bioisoster of the carboxy function. Synthesis, ionization constants, and molecular pharmacological characterization at ionotropic glutamate receptors of compounds related to glutamate and its homologues.
Lolli ML, Giordano C, Pickering DS, Rolando B, Hansen KB, Foti A, Contreras-Sanz A, Amir A, Fruttero R, Gasco A, Nielsen B, Johansen TN. Lolli ML, et al. Among authors: johansen tn. J Med Chem. 2010 May 27;53(10):4110-8. doi: 10.1021/jm1001452. J Med Chem. 2010. PMID: 20408529
Hydroxy-1,2,5-oxadiazolyl moiety as bioisoster of the carboxy function. Synthesis, ionization constants, and pharmacological characterization of gamma-aminobutyric acid (GABA) related compounds.
Lolli ML, Hansen SL, Rolando B, Nielsen B, Wellendorph P, Madsen K, Larsen OM, Kristiansen U, Fruttero R, Gasco A, Johansen TN. Lolli ML, et al. Among authors: johansen tn. J Med Chem. 2006 Jul 13;49(14):4442-6. doi: 10.1021/jm051288b. J Med Chem. 2006. PMID: 16821803
A tetrazolyl-substituted subtype-selective AMPA receptor agonist.
Vogensen SB, Frydenvang K, Greenwood JR, Postorino G, Nielsen B, Pickering DS, Ebert B, Bølcho U, Egebjerg J, Gajhede M, Kastrup JS, Johansen TN, Clausen RP, Krogsgaard-Larsen P. Vogensen SB, et al. Among authors: johansen tn. J Med Chem. 2007 May 17;50(10):2408-14. doi: 10.1021/jm061439q. Epub 2007 Apr 25. J Med Chem. 2007. PMID: 17455929
Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors.
Szymanska E, Frydenvang K, Pickering DS, Krintel C, Nielsen B, Kooshki A, Zachariassen LG, Olsen L, Kastrup JS, Johansen TN. Szymanska E, et al. Among authors: johansen tn. J Med Chem. 2016 Jan 14;59(1):448-61. doi: 10.1021/acs.jmedchem.5b01666. Epub 2015 Dec 22. J Med Chem. 2016. PMID: 26653877
Structural and pharmacological characterization of phenylalanine-based AMPA receptor antagonists at kainate receptors.
Venskutonytė R, Frydenvang K, Valadés EA, Szymańska E, Johansen TN, Kastrup JS, Pickering DS. Venskutonytė R, et al. Among authors: johansen tn. ChemMedChem. 2012 Oct;7(10):1793-8. doi: 10.1002/cmdc.201100599. Epub 2012 Mar 7. ChemMedChem. 2012. PMID: 22407805
A new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure: synthesis, resolution, pharmacology, and crystal structure.
Szymańska E, Frydenvang K, Contreras-Sanz A, Pickering DS, Frola E, Serafimoska Z, Nielsen B, Kastrup JS, Johansen TN. Szymańska E, et al. Among authors: johansen tn. J Med Chem. 2011 Oct 27;54(20):7289-98. doi: 10.1021/jm200862h. Epub 2011 Oct 4. J Med Chem. 2011. PMID: 21923187
3-Substituted phenylalanines as selective AMPA- and kainate receptor ligands.
Szymańska E, Pickering DS, Nielsen B, Johansen TN. Szymańska E, et al. Among authors: johansen tn. Bioorg Med Chem. 2009 Sep 1;17(17):6390-401. doi: 10.1016/j.bmc.2009.07.021. Epub 2009 Jul 16. Bioorg Med Chem. 2009. PMID: 19656686
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